SCHEMBL4715769

SCHEMBL4715769

COc1ccc(S(=O)(=O)N2CCCCC2)cc1COCC(=O)c1ccccn1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 1/20 0.58
MAPK1 P28482 1/20 0.55
SMN1; SMN2 Q16637 3/20 0.51
F2 P00734 1/20 0.51
ALDH1A1 P00352 4/20 0.51
MAPT P10636 3/20 0.50
HTT P42858 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
KDM4E B2RXH2 2/20 0.49
LMNA P02545 1/20 0.49
MDM2 Q00987 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
USP2 O75604 1/20 0.49
HSD17B10 Q99714 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4717827 0.90 MAPK1 (0.61) RXFP1MAPK1SMN1; SMN2F2ALDH1A1
SCHEMBL4713091 0.89 ALDH1A1 (0.54) RXFP1MAPK1SMN1; SMN2ALDH1A1HTT
SCHEMBL8312704 0.88 ALDH1A1 (0.48) RXFP1MAPK1SMN1; SMN2F2ALDH1A1
SCHEMBL4713822 0.81 L3MBTL1 (0.47) MAPK1SMN1; SMN2F2ALDH1A1KDM4E
SCHEMBL5739571 0.81 SMN1; SMN2 (0.52) RXFP1MAPK1SMN1; SMN2ALDH1A1HTT
SCHEMBL4715685 0.79 MCOLN3 (0.51) ALDH1A1MAPTTDP1L3MBTL1
SCHEMBL4716756 0.77 ALDH1A1 (0.55) MAPK1ALDH1A1KDM4EHSD17B10
SCHEMBL4714178 0.77 LMNA (0.57) RXFP1MAPK1SMN1; SMN2ALDH1A1MAPT
SCHEMBL4713433 0.76 SMN1; SMN2 (0.54) MAPK1SMN1; SMN2ALDH1A1MAPTHTT
SCHEMBL8315142 0.76 MAPK1 (0.52) RXFP1MAPK1SMN1; SMN2F2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1615904-B1 SUBSTITUTED BENZOSULPHONAMIDES AS POTENTIATORS OF GLUTAMATE RECEPTORS ASTRAZENECA AB (SE) 2008-02-27 EP claimed
EP-1615904-B1 SUBSTITUTED BENZOSULPHONAMIDES AS POTENTIATORS OF GLUTAMATE RECEPTORS ASTRAZENECA AB (SE) 2008-02-27 EP disclosed
US-20070021606-A1 Therapeutic compounds ASTRAZENECA AB (SE) 2007-01-25 US disclosed
US-20070021606-A1 Therapeutic compounds ASTRAZENECA AB (SE) 2007-01-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070021606-A1 Therapeutic compounds GRIN1, GRIN3A, GRM2 RXFP1 603/4885MAPK1 3513/4885SMN1; SMN2 2089/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.