SCHEMBL4717216

SCHEMBL4717216

NC(=O)c1cc(C[CH]C(=O)N2CCN(c3ccncc3)CC2)cc(Br)c1Cl

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.39
TRPV1 Q8NER1 1/20 0.39
GRM5 P41594 1/20 0.38
CYP17A1 P05093 2/20 0.37
CYP21A2 P08686 2/20 0.37
CYP11B1 P15538 2/20 0.37
AOC3 Q16853 2/20 0.37
F10 P00742 2/20 0.36
CHRM1 P11229 4/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
PARP1 P09874 2/20 0.34
TNKS O95271 1/20 0.34
PARP14 Q460N5 1/20 0.34
HTR4 Q13639 1/20 0.34
F2 P00734 1/20 0.34
PRSS1 P07477 1/20 0.34
ITGB3 P05106 1/20 0.34
ITGA2B P08514 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4862722 0.78 CALCRL (0.38) AOC3PARP1ITGB3ITGA2B
SCHEMBL6802072 0.76 HTR1A (0.39) CYP17A1CYP21A2CYP11B1AOC3F10
SCHEMBL4720815 0.75 L3MBTL3 (0.41)
SCHEMBL4717217 0.68 AKT1 (0.48)
SCHEMBL4851302 0.67 CALCA (0.42) SMN1; SMN2PARP1TNKSPARP14
SCHEMBL4766522 0.67 NAMPT (0.43) SMN1; SMN2
SCHEMBL6601293 0.66 SMN1; SMN2 (0.53) AKR1C3TRPV1SMN1; SMN2
SCHEMBL7010740 0.65 AKT1 (0.49)
SCHEMBL3954177 0.64 CALCRL (0.53)
SCHEMBL7005623 0.63 AKT1 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1558600-B1 SELECTED CGRP ANTAGONISTS, METHOD FOR PRODUCTION AND USE THEREOF AS MEDICAMENT BOEHRINGER INGELHEIM PHARMA (DE) 2008-05-07 EP claimed