SCHEMBL4717751

SCHEMBL4717751

Cc1cc(CC(N)C(=O)N2CCC(N3CCN(CC(F)(F)F)CC3)CC2)ccc1Cl

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MC4R P32245 1/20 0.43
DPP4 P27487 2/20 0.39
CCR5 P51681 2/20 0.39
OPRK1 P41145 2/20 0.39
AKT1 P31749 2/20 0.39
DPP7 Q9UHL4 2/20 0.39
CCR3 P51677 4/20 0.39
OPRD1 P41143 1/20 0.38
AKT2 P31751 1/20 0.38
AKT3 Q9Y243 1/20 0.38
CALCA P06881 2/20 0.37
HDAC8 Q9BY41 1/20 0.36
CHRM2 P08172 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4718742 0.90 MC4R (0.45) MC4RDPP4OPRK1AKT1DPP7
SCHEMBL3314682 0.86 OPRK1 (0.42) MC4RDPP4CCR5OPRK1AKT1
SCHEMBL4722265 0.85 DPP8 (0.47) OPRK1CALCA
SCHEMBL4722468 0.84 AKT1 (0.43) MC4ROPRK1AKT1CCR3OPRD1
SCHEMBL3285190 0.77 OPRK1 (0.44) DPP4CCR5OPRK1OPRD1HDAC8
SCHEMBL3279496 0.76 DPP8 (0.49) OPRK1OPRD1CALCA
SCHEMBL3284873 0.75 L3MBTL3 (0.44) MC4RDPP4CCR5OPRK1OPRD1
SCHEMBL4718313 0.75 OPRK1 (0.42) DPP4CCR5OPRK1DPP7CCR3
SCHEMBL3314171 0.73 DPP8 (0.47) OPRK1CALCA
SCHEMBL4717842 0.73 L3MBTL3 (0.41) DPP4OPRK1AKT1DPP7OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1558600-B1 SELECTED CGRP ANTAGONISTS, METHOD FOR PRODUCTION AND USE THEREOF AS MEDICAMENT BOEHRINGER INGELHEIM PHARMA (DE) 2008-05-07 EP claimed