SCHEMBL4718285

SCHEMBL4718285

COc1cccc(CN2Cc3ccccc3N=C2N)c1OC

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
KDM4E B2RXH2 4/20 0.44
HSP90AA1 P07900 1/20 0.41
HSP90B1 P14625 1/20 0.41
TRAP1 Q12931 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
SIGMAR1 Q99720 1/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 1/20 0.41
ALOX12 P18054 1/20 0.41
MAPK1 P28482 1/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
ATM Q13315 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HSD17B10 Q99714 1/20 0.41
NAMPT P43490 1/20 0.39
BCHE P06276 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3212426 0.99 CA2 (0.45) CA2CA9KDM4EHSP90AA1HSP90B1
SCHEMBL3215576 0.90 SIGMAR1 (0.44) KDM4EMEN1KMT2ASIGMAR1ALDH1A1
Hydrochloric Acid SCHEMBL3210300 0.89 SIGMAR1 (0.43) KDM4EMEN1KMT2ASIGMAR1ALDH1A1
SCHEMBL4714175 0.85 SIGMAR1 (0.44) KDM4ESIGMAR1ALDH1A1HPGDMAPK1
SCHEMBL3197204 0.80 CTSD (0.45) MEN1KMT2ASIGMAR1ALDH1A1CASP1
SCHEMBL3217277 0.80 KDM4E (0.53) KDM4EKMT2ASIGMAR1ALDH1A1MAPK1
SCHEMBL4715614 0.79 CTSD (0.46) KDM4EMEN1KMT2ASIGMAR1ALDH1A1
Acetic Acid SCHEMBL3216929 0.79 SIGMAR1 (0.42) KDM4EMEN1KMT2ASIGMAR1ALDH1A1
SCHEMBL3214965 0.78 SIGMAR1 (0.48) MEN1KMT2ASIGMAR1ACHECTSD
SCHEMBL3222976 0.78 CTSD (0.48) MEN1KMT2ASIGMAR1ALDH1A1BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1917245-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE AS BINDING PARTNERS FOR 5-HT5 RECEPTORS Abbott GmbH & Co. KG (DE) 2008-05-07 EP disclosed
WO-2007022946-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE AS BINDING PARTNERS FOR 5-HT5 RECEPTORS ABBOTT GMBH & CO. KG (DE) 2007-03-01 WO disclosed