SCHEMBL4718989

SCHEMBL4718989

O=C(c1cccnc1F)N1CCN(c2cc(Cl)cc(Cl)c2)CC1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.53
KDM4E B2RXH2 3/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
SMN1; SMN2 Q16637 4/20 0.50
HSD17B10 Q99714 2/20 0.50
USP2 O75604 2/20 0.50
MAPK1 P28482 2/20 0.50
HPGD P15428 1/20 0.50
HTT P42858 3/20 0.49
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
TSHR P16473 3/20 0.48
GAA P10253 1/20 0.47
LMNA P02545 3/20 0.47
MAPT P10636 2/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
ALOX15 P16050 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4722869 0.90 AKR1C3 (0.58) ALDH1A1KDM4EL3MBTL1SMN1; SMN2USP2
SCHEMBL4719103 0.86 ABL1 (0.55) ALDH1A1KDM4EL3MBTL1SMN1; SMN2HSD17B10
SCHEMBL8247070 0.84 SMN1; SMN2 (0.72) ALDH1A1KDM4EL3MBTL1SMN1; SMN2USP2
SCHEMBL8247543 0.84 MEN1 (0.58) ALDH1A1KDM4EL3MBTL1SMN1; SMN2USP2
SCHEMBL4766135 0.82 USP2 (0.57) ALDH1A1KDM4EL3MBTL1SMN1; SMN2USP2
SCHEMBL8240451 0.82 ALDH1A1 (0.60) ALDH1A1KDM4EL3MBTL1SMN1; SMN2HSD17B10
SCHEMBL8250360 0.82 MAPK1 (0.47) ALDH1A1KDM4EL3MBTL1SMN1; SMN2HSD17B10
SCHEMBL4722493 0.80 SMN1; SMN2 (0.54) ALDH1A1KDM4EL3MBTL1SMN1; SMN2USP2
SCHEMBL4722342 0.80 MEN1 (0.71) ALDH1A1KDM4EL3MBTL1SMN1; SMN2HSD17B10
SCHEMBL8246614 0.80 ALDH1A1 (0.62) ALDH1A1SMN1; SMN2HPGDHTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907363-A1 PHENYL SUBSTITUTED PIPERAZINE-DERIVATIVES AS INHIBITORS OF PLAMINOGENIC ACTIVATOR INHIBITORS-I (PAI-I) Bayer HealthCare AG (DE) 2008-04-09 EP disclosed
WO-2007009635-A1 PHENYL SUBSTITUTED PIPERAZINE-DERIVATIVES AS INHIBITORS OF PLAMINOGENIC ACTIVATOR INHIBITORS-I (PAI-I) BAYER HEALTHCARE AG (DE) 2007-01-25 WO disclosed
WO-2007009635-A1 PHENYL SUBSTITUTED PIPERAZINE-DERIVATIVES AS INHIBITORS OF PLAMINOGENIC ACTIVATOR INHIBITORS-I (PAI-I) BAYER HEALTHCARE AG (DE) 2007-01-25 WO disclosed