SCHEMBL4722682

SCHEMBL4722682

O=c1ccc(-c2cccc([N+](=O)[O-])c2)nn1-c1cccc(Cl)c1

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 6/20 0.59
NFE2L2 Q16236 6/20 0.59
MAPT P10636 5/20 0.56
ALDH1A1 P00352 2/20 0.50
TDP1 Q9NUW8 1/20 0.50
RAB9A P51151 4/20 0.48
NPC1 O15118 3/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
HPGD P15428 1/20 0.46
CYP2C19 P33261 1/20 0.46
GFER P55789 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.44
KDM1A O60341 1/20 0.43
IDO1 P14902 1/20 0.43
GSK3A P49840 1/20 0.43
GSK3B P49841 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4720647 0.92 KEAP1 (0.55) KEAP1NFE2L2MAPTALDH1A1RAB9A
SCHEMBL4722007 0.90 KEAP1 (0.50) KEAP1NFE2L2MAPTALDH1A1TDP1
SCHEMBL4724761 0.89 KEAP1 (0.56) KEAP1NFE2L2MAPTALDH1A1TDP1
SCHEMBL4722872 0.87 KEAP1 (0.60) KEAP1NFE2L2MAPTALDH1A1RAB9A
SCHEMBL4720269 0.86 KEAP1 (0.48) KEAP1NFE2L2MAPTRAB9ANPC1
SCHEMBL4722720 0.83 KEAP1 (0.49) KEAP1NFE2L2MAPTALDH1A1TDP1
SCHEMBL4720939 0.78 MAPT (0.51) KEAP1NFE2L2MAPTALDH1A1RAB9A
SCHEMBL4721400 0.78 KEAP1 (0.44) KEAP1NFE2L2MAPTALDH1A1TDP1
SCHEMBL4721008 0.77 MAPT (0.49) KEAP1NFE2L2MAPTALDH1A1TDP1
SCHEMBL4724756 0.77 NPSR1 (0.47) KEAP1NFE2L2MAPTTDP1GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP claimed
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed