SCHEMBL4722007

SCHEMBL4722007

O=c1ccc(-c2cccc([N+](=O)[O-])c2)nn1-c1ccc(Cl)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 3/20 0.50
NFE2L2 Q16236 3/20 0.50
MAPT P10636 4/20 0.48
RAB9A P51151 1/20 0.48
PSD A5PKW4 1/20 0.48
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CNR1 P21554 1/20 0.44
ALDH1A1 P00352 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
IDO1 P14902 1/20 0.43
GABRA1 P14867 2/20 0.43
GABRB2 P47870 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
GABRP O00591 1/20 0.42
GABRD O14764 1/20 0.42
GABRB1 P18505 1/20 0.42
GABRG2 P18507 1/20 0.42
GABRB3 P28472 1/20 0.42
GABRA5 P31644 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4720269 0.91 KEAP1 (0.48) KEAP1NFE2L2MAPTRAB9ACA1
SCHEMBL4722682 0.90 KEAP1 (0.59) KEAP1NFE2L2MAPTRAB9AALDH1A1
SCHEMBL4724761 0.89 KEAP1 (0.56) KEAP1NFE2L2MAPTRAB9AALDH1A1
SCHEMBL4722720 0.88 KEAP1 (0.49) KEAP1NFE2L2MAPTRAB9ACA1
SCHEMBL4720647 0.87 KEAP1 (0.55) KEAP1NFE2L2MAPTRAB9AALDH1A1
SCHEMBL4722872 0.82 KEAP1 (0.60) KEAP1NFE2L2MAPTRAB9AALDH1A1
SCHEMBL8422149 0.78 PTGS2 (0.66)
SCHEMBL8121830 0.78 PTGS2 (0.66) SMN1; SMN2
SCHEMBL4720939 0.78 MAPT (0.51) KEAP1NFE2L2MAPTRAB9AALDH1A1
SCHEMBL4721400 0.78 KEAP1 (0.44) KEAP1NFE2L2MAPTRAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP claimed
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed