SCHEMBL4722720

SCHEMBL4722720

Cc1ccc(-n2nc(-c3cccc([N+](=O)[O-])c3)ccc2=O)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 3/20 0.49
NFE2L2 Q16236 3/20 0.49
MAPT P10636 7/20 0.48
ALDH1A1 P00352 4/20 0.48
NPC1 O15118 4/20 0.48
RAB9A P51151 4/20 0.48
GAA P10253 1/20 0.48
HPGD P15428 1/20 0.48
CASP3 P42574 1/20 0.48
HTT P42858 1/20 0.48
SENP7 Q9BQF6 1/20 0.48
SMN1; SMN2 Q16637 4/20 0.47
PKM P14618 1/20 0.47
MEN1 O00255 1/20 0.45
GFER P55789 1/20 0.45
KMT2A Q03164 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
MAOB P27338 1/20 0.45
THRB P10828 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4720269 0.91 KEAP1 (0.48) KEAP1NFE2L2MAPTNPC1RAB9A
SCHEMBL4722872 0.89 KEAP1 (0.60) KEAP1NFE2L2MAPTALDH1A1NPC1
SCHEMBL4724761 0.89 KEAP1 (0.56) KEAP1NFE2L2MAPTALDH1A1NPC1
SCHEMBL4722007 0.88 KEAP1 (0.50) KEAP1NFE2L2MAPTALDH1A1RAB9A
SCHEMBL4720647 0.87 KEAP1 (0.55) KEAP1NFE2L2MAPTALDH1A1NPC1
SCHEMBL4722682 0.83 KEAP1 (0.59) KEAP1NFE2L2MAPTALDH1A1NPC1
SCHEMBL4721008 0.82 MAPT (0.49) KEAP1NFE2L2MAPTALDH1A1NPC1
SCHEMBL4721400 0.78 KEAP1 (0.44) KEAP1NFE2L2MAPTALDH1A1NPC1
SCHEMBL4720939 0.78 MAPT (0.51) KEAP1NFE2L2MAPTALDH1A1NPC1
SCHEMBL4458062 0.74 CASP3 (0.53) KEAP1NFE2L2MAPTALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP claimed
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed