SCHEMBL4723154

SCHEMBL4723154

COc1cc(OC)cc(-c2cn(-c3cc(Br)ccc3C(F)(F)F)c(=O)c3c2CCN3)c1

nearest known ligand 0.32

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AKR1B10 O60218 1/20 0.32
AKR1C4 P17516 1/20 0.32
AKR1C3 P42330 1/20 0.32
AKR1C2 P52895 1/20 0.32
AKR1C1 Q04828 1/20 0.32
CRHR1 P34998 1/20 0.31
LRRK2 Q5S007 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4719266 0.81 LRRK2 (0.33) CRHR1LRRK2
SCHEMBL4719047 0.78 ITGB2 (0.40)
SCHEMBL4719042 0.78 ITGB2 (0.40)
SCHEMBL4722849 0.77 BRD4 (0.45)
SCHEMBL4722066 0.76
SCHEMBL14101952 0.76 AKR1B10 (0.32) AKR1B10AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL4720890 0.76 EGFR (0.33)
SCHEMBL4720875 0.75 BRD4 (0.37)
SCHEMBL4721608 0.73 AKR1B10 (0.33) AKR1B10AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL4719016 0.71 AKR1B10 (0.33) AKR1B10AKR1C4AKR1C3AKR1C2AKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed