SCHEMBL4720875

SCHEMBL4720875

COc1cc(OC)cc(-c2cn(-c3cc(Br)ccc3C(F)(F)F)c(=O)c3c2CCN3C(=O)c2ccccc2)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.37
LMNA P02545 5/20 0.37
PDCD1 Q15116 6/20 0.36
CD274 Q9NZQ7 6/20 0.36
ALDH1A1 P00352 2/20 0.35
MAPT P10636 1/20 0.35
ALOX15 P16050 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
TSHR P16473 1/20 0.35
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
KDM4E B2RXH2 2/20 0.33
KMT2A Q03164 2/20 0.33
TUBB4A P04350 1/20 0.33
TUBB P07437 1/20 0.33
TUBA3C P0DPH7 1/20 0.33
TUBA1B P68363 1/20 0.33
TUBA4A P68366 1/20 0.33
TUBB4B P68371 1/20 0.33
TUBB3 Q13509 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4722418 0.79 PDCD1 (0.32) LMNAPDCD1CD274
SCHEMBL4723154 0.75 AKR1B10 (0.32)
SCHEMBL4719251 0.75 ACVR1 (0.35)
SCHEMBL4719937 0.75 ACVR1 (0.32)
SCHEMBL4722741 0.72 UCHL1 (0.38) LMNAMAPTKMT2AMEN1
SCHEMBL4722281 0.71 LIPG (0.38) NOTUM
SCHEMBL4722284 0.71 LIPG (0.38) NOTUM
SCHEMBL4719016 0.71 AKR1B10 (0.33) ALDH1A1TDP1KDM4E
SCHEMBL14101950 0.70 UCHL1 (0.37) BRD4KMT2AMEN1
SCHEMBL4720890 0.70 EGFR (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed