SCHEMBL4723702

SCHEMBL4723702

COc1cc(OC)cc(-c2nn(-c3cc(N4CCN(C(C)=O)CC4)ccc3C(F)(F)F)c(=O)c3c2CCC3)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 13/20 0.40
MAPT P10636 3/20 0.38
CYP2C9 P11712 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
USP2 O75604 2/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
KMT2A Q03164 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
LMNA P02545 2/20 0.36
GAA P10253 1/20 0.36
MAPK1 P28482 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4720515 0.91 LMNA (0.38) ALKMAPTCYP2C9HDAC6USP2
SCHEMBL4724195 0.91 F10 (0.42) MAPTALDH1A1PDE4APDE4BPDE4C
SCHEMBL4724509 0.91 PDE4A (0.41) MAPTPDE4APDE4BPDE4CPDE4D
SCHEMBL4722495 0.90 F10 (0.44) MAPTCYP2C9ALDH1A1NPSR1PDE4A
SCHEMBL4722762 0.88 F10 (0.39) MAPTCYP2C9USP2MEN1ALDH1A1
SCHEMBL4721093 0.88 PDE4A (0.37) MAPTPDE4APDE4BPDE4CPDE4D
SCHEMBL4722548 0.86 PDE4A (0.37) PDE4APDE4BPDE4CPDE4D
SCHEMBL14101702 0.86 F10 (0.40) MAPTALDH1A1NPSR1PDE4APDE4B
SCHEMBL4721967 0.86 PDE4A (0.38) PDE4APDE4BPDE4CPDE4D
SCHEMBL4722276 0.85 UGCG (0.36) PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed