SCHEMBL4723245

SCHEMBL4723245

Nc1ccccc1-n1nc(-c2cccc(Cl)c2)ccc1=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.51
GAA P10253 3/20 0.51
MAPT P10636 3/20 0.51
MEN1 O00255 2/20 0.51
LMNA P02545 2/20 0.51
KMT2A Q03164 2/20 0.51
TDP1 Q9NUW8 2/20 0.51
L3MBTL1 Q9Y468 2/20 0.51
TP53 P04637 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
HDAC1 Q13547 1/20 0.49
MAPK1 P28482 1/20 0.48
ADORA2A P29274 1/20 0.44
ADORA1 P30542 1/20 0.44
PARP1 P09874 1/20 0.42
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
ATM Q13315 1/20 0.41
TSHR P16473 1/20 0.40
DPP4 P27487 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4723906 0.81 HDAC1 (0.51) KDM4ELMNATDP1NPSR1HDAC1
SCHEMBL4724756 0.80 NPSR1 (0.47) KDM4EGAAMAPTMEN1LMNA
SCHEMBL4054250 0.70 KDM4E (0.55) KDM4EGAAMAPTMEN1KMT2A
SCHEMBL2470246 0.68 HDAC1 (0.59) KDM4EGAAMAPTMEN1LMNA
SCHEMBL4722682 0.68 KEAP1 (0.59) MAPTTDP1NPC1RAB9A
SCHEMBL28073914 0.67 GAA (0.46) KDM4EGAAMAPTMEN1LMNA
SCHEMBL10686701 0.67 TSHR (0.56) KDM4EGAAMAPTMEN1LMNA
SCHEMBL4055321 0.67 HDAC1 (0.45) KDM4EGAAMAPTMEN1LMNA
SCHEMBL4765637 0.66 MAPT (0.48) KDM4EGAAMAPTMEN1LMNA
SCHEMBL8420106 0.66 PTGS2 (0.48) PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP claimed
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed