Pyrrolidine

Pyrrolidine

SCHEMBL4724716

C1CCNC1.FC(F)(F)c1nc2ccccc2[nH]1

nearest known ligand 0.77

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 4/20 0.77
ALDH1A1 P00352 7/20 0.47
KDM4E B2RXH2 5/20 0.47
MAPT P10636 5/20 0.47
PKM P14618 3/20 0.47
GAA P10253 2/20 0.47
KHK P50053 1/20 0.47
HSD17B10 Q99714 2/20 0.46
HPGD P15428 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
ALOX15 P16050 1/20 0.46
CYP2C19 P33261 1/20 0.46
HTR3A P46098 1/20 0.46
POLB P06746 4/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
THRB P10828 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29353981 0.88 NPSR1 (1.00) NPSR1ALDH1A1KDM4EMAPTPKM
SCHEMBL10295 0.88 NPSR1 (1.00) NPSR1ALDH1A1KDM4EMAPTPKM
SCHEMBL27974001 0.83 NPSR1 (0.89) NPSR1ALDH1A1KDM4EMAPTPKM
Diphenylether SCHEMBL4184182 0.77 NPSR1 (0.77) NPSR1ALDH1A1KDM4EMAPTPKM
SCHEMBL4374246 0.77 NPSR1 (0.78) NPSR1ALDH1A1KDM4EMAPTPKM
SCHEMBL27840000 0.75 NPSR1 (0.75) NPSR1ALDH1A1KDM4EMAPTPKM
SCHEMBL9960528 0.75 NPSR1 (0.75) NPSR1ALDH1A1KDM4EMAPTPKM
Pyrrolidine SCHEMBL4830345 0.75 RAB9A (0.54) NPSR1ALDH1A1KDM4EPKMGAA
SCHEMBL23854433 0.74 NPSR1 (0.72) NPSR1ALDH1A1KDM4EMAPTPKM
SCHEMBL5015526 0.74 NPSR1 (0.72) NPSR1ALDH1A1KDM4EMAPTPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1994022-A2 N-SUBSTITUTED-AZACYCLYLAMINES AS HISTAMINE-3 ANTAGONISTS Wyeth a Corporation of the State of Delaware (US) 2008-11-26 EP disclosed
WO-2007108936-A2 N-SUBSTITUTED-AZACYCLYLAMINES AS HISTAMINE-3 ANTAGONISTS WYETH (US) 2007-09-27 WO disclosed