SCHEMBL4725669

SCHEMBL4725669

N#Cc1cc(C#N)cc(N2CCOCC2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.51
LMNA P02545 2/20 0.51
MAPT P10636 2/20 0.51
HTT P42858 2/20 0.51
NSD2 O96028 1/20 0.51
TSHR P16473 1/20 0.51
CASP1 P29466 1/20 0.51
CASP7 P55210 1/20 0.51
CASP6 P55212 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
MAPK1 P28482 1/20 0.46
AR P10275 1/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
PRKDC P78527 3/20 0.43
DRD2 P14416 1/20 0.43
DRD3 P35462 1/20 0.43
TP53 P04637 1/20 0.43
AKT1 P31749 1/20 0.42
PIK3CA P42336 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31703179 0.88 MAPK1 (0.47) KDM4ELMNAMAPTHTTNSD2
SCHEMBL594313 0.88 KDM4E (0.49) KDM4ELMNAMAPTHTTNSD2
SCHEMBL31703324 0.88 KDM4E (0.45) KDM4ELMNAMAPTHTTNSD2
SCHEMBL4758228 0.88 MAPK1 (0.47) KDM4ELMNAMAPTHTTNSD2
SCHEMBL3760756 0.88 KDM4E (0.45) KDM4ELMNAMAPTHTTNSD2
SCHEMBL4434635 0.88 KDM4E (0.45) KDM4ELMNAMAPTHTTNSD2
SCHEMBL4757023 0.88 LMNA (0.49) KDM4ELMNAMAPTHTTNSD2
SCHEMBL3530448 0.84 ADRB1 (0.49) KDM4ELMNAMAPTHTTNSD2
SCHEMBL14293712 0.82 KMO (0.56) KDM4ELMNAMAPTHTTNSD2
SCHEMBL3783100 0.82 DRD2 (0.68) KDM4ELMNAMAPTHTTNSD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021388-A1 HETEROARYL DERIVATIVES AS CYTOKINE INHIBITORS KEMIA, INC. (US) 2008-02-21 WO disclosed
WO-2008021388-A1 HETEROARYL DERIVATIVES AS CYTOKINE INHIBITORS KEMIA, INC. (US) 2008-02-21 WO disclosed
WO-2007075896-A2 HETEROCYCLIC CYTOKINE INHIBITORS KEMIA, INC. (US) 2007-07-05 WO disclosed
WO-2007075896-A2 HETEROCYCLIC CYTOKINE INHIBITORS KEMIA, INC. (US) 2007-07-05 WO disclosed