SCHEMBL4728357

SCHEMBL4728357

Cc1cc(OCc2ccc(-c3ccc(C(F)(F)F)nc3)nc2C)ccc1CCCCn1ccnn1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 1/20 0.37
MINK1 Q8N4C8 1/20 0.37
PPARD Q03181 6/20 0.36
PPARG P37231 2/20 0.36
PPARA Q07869 2/20 0.36
TRPV3 Q8NET8 4/20 0.33
GRM2 Q14416 1/20 0.33
FFAR1 O14842 1/20 0.33
FFAR4 Q5NUL3 1/20 0.33
ATP4A P20648 1/20 0.33
ATP4B P51164 1/20 0.33
GRM5 P41594 1/20 0.32
MAOA P21397 1/20 0.31
PTGES O14684 1/20 0.30
ALOX5AP P20292 1/20 0.30
RXFP1 Q9HBX9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4780494 0.90 ERBB2 (0.46) ERBB2MINK1PPARDPPARGPPARA
SCHEMBL4600061 0.89 ERBB2 (0.45) ERBB2MINK1PPARDPPARGPPARA
SCHEMBL4780947 0.88 ATP4A (0.34) ERBB2MINK1PPARDPPARGPPARA
SCHEMBL4599602 0.88 PPARD (0.39) ERBB2MINK1PPARDPPARGPPARA
SCHEMBL4728989 0.87 TRPV3 (0.34) PPARDPPARGPPARATRPV3GRM2
SCHEMBL4782623 0.87 PPARD (0.34) PPARDPPARGPPARATRPV3GRM2
SCHEMBL4591853 0.87 ATP4A (0.37) ERBB2MINK1PPARDPPARGPPARA
SCHEMBL4600066 0.86 ERBB2 (0.41) ERBB2MINK1PPARDPPARGPPARA
SCHEMBL4726101 0.86 TRPV3 (0.32) ERBB2MINK1TRPV3GRM2ATP4A
SCHEMBL4599860 0.85 ATP4A (0.37) ERBB2MINK1PPARDPPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008034579-A1 2-HETEROCYCLYL-5-PHENOXYMETHYLPYRIDINE DERIVATIVES AS ANTICANCER AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2008-03-27 WO disclosed