SCHEMBL4728989

SCHEMBL4728989

Cc1cc(OCc2ccc(-c3ccc(C(F)(F)F)nc3)nc2C)ccc1C(O)CCCn1ccnn1

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TRPV3 Q8NET8 10/20 0.34
SCN9A Q15858 1/20 0.33
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33
APH1A Q96BI3 1/20 0.33
PSENEN Q9NZ42 1/20 0.33
MAOA P21397 2/20 0.32
GRM2 Q14416 1/20 0.32
PTGES O14684 1/20 0.32
PPARD Q03181 3/20 0.32
PPARG P37231 1/20 0.32
PPARA Q07869 1/20 0.32
ATP4A P20648 1/20 0.31
ATP4B P51164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4726101 0.91 TRPV3 (0.32) TRPV3PSEN1PSEN2APH1BNCSTN
SCHEMBL4732040 0.89 TRPV3 (0.35) TRPV3SCN9APSEN1PSEN2APH1B
SCHEMBL4730017 0.89 PSEN1 (0.34) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL4728357 0.87 ERBB2 (0.37) TRPV3MAOAGRM2PTGESPPARD
SCHEMBL4782623 0.85 PPARD (0.34) TRPV3MAOAGRM2PTGESPPARD
SCHEMBL4730718 0.83 GRM2 (0.34) TRPV3PSEN1PSEN2APH1BNCSTN
SCHEMBL4784127 0.83 PPARD (0.33) TRPV3MAOAGRM2PTGESPPARD
SCHEMBL4780494 0.82 ERBB2 (0.46) TRPV3GRM2PTGESPPARDPPARG
SCHEMBL4728771 0.82 MMP1 (0.34) TRPV3GRM2PPARDATP4AATP4B
SCHEMBL4782456 0.81 PPARD (0.36) TRPV3GRM2PPARDPPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008034579-A1 2-HETEROCYCLYL-5-PHENOXYMETHYLPYRIDINE DERIVATIVES AS ANTICANCER AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2008-03-27 WO claimed
WO-2008034579-A1 2-HETEROCYCLYL-5-PHENOXYMETHYLPYRIDINE DERIVATIVES AS ANTICANCER AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2008-03-27 WO disclosed