SCHEMBL4780494

SCHEMBL4780494

Cc1nc(-c2ccc(C(F)(F)F)nc2)ccc1COc1ccc(CCCCn2ccnn2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 1/20 0.46
MINK1 Q8N4C8 1/20 0.46
GRM2 Q14416 1/20 0.37
ATP4A P20648 1/20 0.37
ATP4B P51164 1/20 0.37
GRM5 P41594 1/20 0.35
RXRA P19793 3/20 0.34
NR1H2 P55055 3/20 0.34
NR1H3 Q13133 1/20 0.33
PPARD Q03181 3/20 0.33
PPARG P37231 2/20 0.33
PPARA Q07869 2/20 0.33
FFAR4 Q5NUL3 2/20 0.33
PLAAT3 P53816 1/20 0.33
PLAAT5 Q96KN8 1/20 0.33
PLAAT2 Q9NWW9 1/20 0.33
PLAAT4 Q9UL19 1/20 0.33
TRPV3 Q8NET8 3/20 0.33
FFAR1 O14842 1/20 0.32
THRB P10828 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4728357 0.90 ERBB2 (0.37) ERBB2MINK1GRM2ATP4AATP4B
SCHEMBL4600322 0.89 ERBB2 (0.56) ERBB2MINK1ATP4AATP4BRXRA
SCHEMBL4602065 0.87 ERBB2 (0.46) ERBB2MINK1GRM2ATP4AATP4B
SCHEMBL4726900 0.87 ERBB2 (0.41) ERBB2MINK1GRM2ATP4AATP4B
SCHEMBL4732040 0.86 TRPV3 (0.35) ERBB2MINK1GRM2ATP4AATP4B
SCHEMBL4728771 0.86 MMP1 (0.34) ERBB2MINK1GRM2ATP4AATP4B
SCHEMBL4599664 0.86 ERBB2 (0.44) ERBB2MINK1ATP4AATP4BPPARD
SCHEMBL4599925 0.85 ERBB2 (0.50) ERBB2MINK1ATP4AATP4BRXRA
SCHEMBL4730718 0.85 GRM2 (0.34) ERBB2MINK1GRM2ATP4AATP4B
SCHEMBL4599913 0.84 ERBB2 (0.42) ERBB2MINK1ATP4AATP4BFFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008034579-A1 2-HETEROCYCLYL-5-PHENOXYMETHYLPYRIDINE DERIVATIVES AS ANTICANCER AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2008-03-27 WO claimed
WO-2008034579-A1 2-HETEROCYCLYL-5-PHENOXYMETHYLPYRIDINE DERIVATIVES AS ANTICANCER AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2008-03-27 WO disclosed