SCHEMBL4729100

SCHEMBL4729100

CC(C)(C)[Si](C)(C)OCc1ccc(-c2csc(CI)n2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 8/20 0.43
L3MBTL1 Q9Y468 6/20 0.43
NPC1 O15118 6/20 0.43
CASP3 P42574 1/20 0.43
SENP8 Q96LD8 1/20 0.43
SENP7 Q9BQF6 1/20 0.43
SENP6 Q9GZR1 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
MAPT P10636 7/20 0.42
ALDH1A1 P00352 6/20 0.41
MEN1 O00255 6/20 0.40
KMT2A Q03164 5/20 0.40
KDM4E B2RXH2 3/20 0.40
POLB P06746 3/20 0.40
PKM P14618 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
OPRK1 P41145 1/20 0.40
GAA P10253 2/20 0.39
APEX1 P27695 1/20 0.39
RECQL P46063 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4729130 0.87 RAB9A (0.45) RAB9AL3MBTL1NPC1CASP3SENP8
SCHEMBL5221804 0.81 IDO1 (0.35)
SCHEMBL4728570 0.81 RAB9A (0.69) RAB9AL3MBTL1NPC1CASP3SENP8
SCHEMBL3426875 0.80 AGXT (0.32)
SCHEMBL16319093 0.76 L3MBTL1 (0.65) RAB9AL3MBTL1NPC1CASP3SENP8
SCHEMBL4730043 0.73 PTPN1 (0.41) RAB9AL3MBTL1NPC1CASP3SENP8
SCHEMBL219652 0.72 RAB9A (0.44) RAB9AL3MBTL1NPC1CASP3SENP8
SCHEMBL28129052 0.71 DUT (0.33)
SCHEMBL9033464 0.71 CYP17A1 (0.46) L3MBTL1TDP1LTA4H
SCHEMBL6615170 0.70 BACE1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008033455-A2 BIPHENYL AND HETEROARYL PHENYL DERIVATIVES AS PROTEIN TYROSINE PHOSPHATASES INHIBITORS THE INSTITUTES FOR PHARMACEUTICAL DISCOVERY, LLC (US) 2008-03-20 WO disclosed