SCHEMBL4729403

SCHEMBL4729403

COc1cc(N)c2nc(C(C)C)ccc2c1OC

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC10A2 Q12908 1/20 0.38
NSD2 O96028 1/20 0.38
CASP6 P55212 1/20 0.38
G6PD P11413 1/20 0.38
PDE5A O76074 1/20 0.37
DHFR P00374 1/20 0.37
TYMS P04818 1/20 0.37
TSHR P16473 3/20 0.35
ALDH1A1 P00352 2/20 0.35
CYP3A4 P08684 2/20 0.35
HSD17B10 Q99714 2/20 0.35
TDP1 Q9NUW8 1/20 0.35
MAOA P21397 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4727095 0.87 NSD2 (0.38) NSD2CASP6G6PDDHFRTSHR
SCHEMBL4726183 0.77 TUBB4A (0.40) TYMSALDH1A1CYP3A4HSD17B10TDP1
SCHEMBL4727819 0.77 NSD2 (0.38) NSD2CASP6G6PDPDE5ADHFR
SCHEMBL4726086 0.73 MEN1 (0.48) SLC10A2NSD2CASP6PDE5ATSHR
SCHEMBL5080779 0.73 HSP90AA1 (0.53) NSD2CASP6ALDH1A1CYP3A4MAOA
SCHEMBL28248381 0.72 NOS3 (0.37) TSHRALDH1A1HSD17B10TDP1KDM4E
SCHEMBL4780864 0.71 CYP1A2 (0.33) NSD2CASP6G6PDALDH1A1CYP3A4
SCHEMBL5083088 0.71 TUBB4A (0.39) NSD2CASP6G6PDTSHRALDH1A1
SCHEMBL423613 0.71 CASP6 (0.70) NSD2CASP6G6PDPDE5AALDH1A1
SCHEMBL25911059 0.69 TLR8 (0.42) SLC10A2KDM4EIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021210-A2 METHODS AND COMPOSITIONS FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS COMBINATORX, INCORPORATED (US) 2008-02-21 WO disclosed
US-20080044390-A1 Methods and compositions for the treatment of neurodegenerative disorders CHDI, INCORPORATED 2008-02-21 US disclosed
US-6979740-B2 Process for preparation of ring-substituted 8-aminoquinoline analogs as antimalarial agents NATIONAL INSTITUTE OF PHARMACEUTICAL EDUCATION AND RESEARCH (IN) 2005-12-27 US disclosed
US-20040192724-A1 Process for preparation of ring-substituted 8-aminoquinoline analogs as antimalarial agents NATIONAL INSTITUTE OF PHARMACEUTICAL EDUCATION AND RESEARCH DEPARTMENT OF PHARMACEUTICAL TECHNOLOGY (IN) 2004-09-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040192724-A1 Process for preparation of ring-substituted 8-aminoquinoline analogs as antimalarial agents QDPR, SLC11A2, CYP2C8 SLC10A2 4736/4885NSD2 2330/4885CASP6 612/4885
US-20080044390-A1 Methods and compositions for the treatment of neurodegenerative disorders HTT, SNCA, NLN SLC10A2 3148/4885NSD2 1540/4885CASP6 897/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.