SCHEMBL4730378

SCHEMBL4730378

Cc1nc(NC2CCCCC2)cc(S(=O)(=O)N2CCOCC2)c1C

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.51
RAB9A P51151 3/20 0.50
NPC1 O15118 2/20 0.50
ALDH1A1 P00352 4/20 0.48
GAA P10253 3/20 0.46
KDM4E B2RXH2 2/20 0.46
NPSR1 Q6W5P4 2/20 0.46
HPGD P15428 1/20 0.46
OPRM1 P35372 1/20 0.46
OPRD1 P41143 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
KMT2A Q03164 2/20 0.45
CNR1 P21554 5/20 0.45
CNR2 P34972 5/20 0.45
TSHR P16473 2/20 0.45
PKM P14618 1/20 0.43
USP2 O75604 1/20 0.42
HSD17B10 Q99714 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4734532 0.82 NPC1 (0.55) LMNARAB9ANPC1ALDH1A1GAA
SCHEMBL4782358 0.77 CNR2 (0.52) ALDH1A1CNR1CNR2PKM
SCHEMBL4732719 0.74 PKM (0.51) LMNAALDH1A1GAANPSR1SMN1; SMN2
SCHEMBL4733274 0.73 CNR2 (0.69) CNR1CNR2
SCHEMBL5624844 0.67 NPC1 (1.00) RAB9ANPC1ALDH1A1GAAKDM4E
SCHEMBL17749369 0.65 LMNA (0.66) LMNAALDH1A1GAAKDM4ENPSR1
SCHEMBL15834046 0.64 HRH4 (0.48) RAB9ANPC1ALDH1A1GAAKDM4E
SCHEMBL17749349 0.63 WNK1 (0.62) LMNAALDH1A1GAAKDM4EHPGD
SCHEMBL5253649 0.62 CTSK (0.58) ALDH1A1KDM4EHSD17B10
SCHEMBL17300713 0.62 HRH4 (0.45) ALDH1A1GAAKDM4EHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008063625-A2 PYRIDINE COMPOUNDS AND METHODS OF THEIR USE ADOLOR CORPORATION (US) 2008-05-29 WO claimed
WO-2008063625-A2 PYRIDINE COMPOUNDS AND METHODS OF THEIR USE ADOLOR CORPORATION (US) 2008-05-29 WO disclosed