SCHEMBL4730798

SCHEMBL4730798

CN(C)C(=S)Oc1ccccc1C(C)(C)C

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.47
ATM Q13315 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.44
ALDH1A1 P00352 4/20 0.44
KDM4E B2RXH2 3/20 0.44
BCHE P06276 1/20 0.42
TSHR P16473 1/20 0.39
GAA P10253 1/20 0.38
KMT2A Q03164 1/20 0.38
RXRA P19793 1/20 0.38
RXRB P28702 1/20 0.38
RXRG P48443 1/20 0.38
NISCH Q9Y2I1 1/20 0.37
MAPT P10636 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CA2 P00918 1/20 0.36
TRPV1 Q8NER1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9351809 0.84 ADRA2A (0.40) L3MBTL1ALDH1A1KMT2ARXRARXRB
SCHEMBL6872602 0.78 TDP1 (0.50) TDP1ATMALDH1A1KDM4EBCHE
SCHEMBL13158912 0.76 ALDH1A1 (0.39) TDP1ATML3MBTL1ALDH1A1KDM4E
SCHEMBL24813703 0.76 TP53 (0.48) TDP1ATML3MBTL1ALDH1A1KDM4E
SCHEMBL10584699 0.75 TDP1 (0.54) TDP1ATMALDH1A1KDM4EBCHE
SCHEMBL22829872 0.74 FABP7 (0.37) L3MBTL1ALDH1A1BCHETSHRMAPT
SCHEMBL27269441 0.74 NR1I2 (0.52) TDP1ATMALDH1A1KDM4EBCHE
SCHEMBL10932562 0.74 TDP1 (0.36) TDP1ATMALDH1A1KDM4EBCHE
SCHEMBL47807 0.73 TDP1 (0.62) TDP1ATMALDH1A1KDM4EBCHE
SCHEMBL30134334 0.73 TDP1 (0.62) TDP1ATMALDH1A1KDM4EBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008061006-A1 SUBSTITUTED INDAN-2-YL, TETRAHYDRONAPHTHALEN-2-YL, OR DIHYDR0-2H-CHR0MEN-3-YL ARYLSULFONAMIDES AND METHODS OF THEIR USE WYETH (US) 2008-05-22 WO disclosed
US-5359065-A Reacting a bromo aromatic compound with an excess of silylating agent; forming metallized intermediate; quenching EASTMAN KODAK COMPANY (US) 1994-10-25 US disclosed