SCHEMBL473100

SCHEMBL473100

CCCCOC(=O)NNc1ccccc1C

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 5/20 0.59
GAA P10253 6/20 0.58
CYP1A2 P05177 3/20 0.57
CYP2C19 P33261 3/20 0.57
SMN1; SMN2 Q16637 3/20 0.57
TDP1 Q9NUW8 2/20 0.54
KDM4E B2RXH2 1/20 0.54
ALDH1A1 P00352 2/20 0.50
RAB9A P51151 4/20 0.48
NPC1 O15118 3/20 0.48
TSHR P16473 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
HPGD P15428 3/20 0.46
CYP2C9 P11712 2/20 0.46
POLB P06746 1/20 0.44
MAPT P10636 1/20 0.44
LMNA P02545 1/20 0.44
DHODH Q02127 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL474568 0.94 P2RX7 (0.64) P2RX7GAACYP1A2CYP2C19SMN1; SMN2
SCHEMBL13506223 0.85 SMN1; SMN2 (0.68) CYP1A2CYP2C19SMN1; SMN2KDM4EALDH1A1
SCHEMBL2234416 0.83 GAA (0.59) GAACYP1A2CYP2C19SMN1; SMN2TDP1
SCHEMBL29290659 0.81 SMN1; SMN2 (0.62) P2RX7CYP1A2CYP2C19SMN1; SMN2ALDH1A1
SCHEMBL1625209 0.80 GAA (0.71) GAACYP1A2CYP2C19SMN1; SMN2TDP1
SCHEMBL5923508 0.77 P2RX7 (0.88) P2RX7GAATDP1KDM4EALDH1A1
O-Xylene SCHEMBL27872004 0.77 ALDH1A1 (0.53) CYP1A2CYP2C19SMN1; SMN2TDP1KDM4E
SCHEMBL1956240 0.77 NLRP3 (0.66) GAACYP1A2CYP2C19SMN1; SMN2TDP1
SCHEMBL473102 0.76 SMN1; SMN2 (0.56) GAACYP1A2CYP2C19SMN1; SMN2KDM4E
SCHEMBL5923449 0.76 P2RX7 (0.97) P2RX7GAATDP1KDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2527297-B1 PROCESS FOR PRODUCTION OF ZINC TOLUENESULFONATE, ZINC TOLUENESULFONATE, AND PROCESS FOR PRODUCTION OF CARBAMATE MITSUI CHEMICALS INC (JP) 2018-11-21 EP disclosed
EP-2412703-B1 URETHANE COMPOUND AND PROCESS FOR PRODUCTION THEREOF, AND ISOCYANATE AND PROCESS FOR PRODUCTION THEREOF MITSUI CHEMICALS INC (JP) 2016-06-29 EP disclosed
EP-2518044-B1 METHOD FOR TREATMENT OF ISOCYANATE RESIDUE, AND METHOD FOR TREATMENT OF CARBONATE MITSUI CHEMICALS INC (JP) 2016-04-13 EP disclosed
US-9150502-B2 Urethane compound and method for producing the same, and isocyanate and method for producing the same MITSUI CHEMICALS, INC. (JP) 2015-10-06 US disclosed
US-9000219-B2 Method for treatment of isocyanate residue, and method for treatment of carbonate MITSUI CHEMICALS, INC. (JP) 2015-04-07 US disclosed
US-8664420-B2 Process for production of zinc toluenesulfonate, zinc toluenesulfonate, and process for production of carbamate MITSUI CHEMICALS, INC. (JP) 2014-03-04 US disclosed
EP-2518044-A1 METHOD FOR TREATMENT OF ISOCYANATE RESIDUE, AND METHOD FOR TREATMENT OF CARBONATE Mitsui Chemicals, Inc. (JP) 2012-10-31 EP disclosed
US-20120271067-A1 METHOD FOR TREATMENT OF ISOCYANATE RESIDUE, AND METHOD FOR TREATMENT OF CARBONATE MITSUI CHEMICALS, INC. 2012-10-25 US disclosed
US-20120259134-A1 PROCESS FOR PRODUCTION OF ZINC TOLUENESULFONATE, ZINC TOLUENESULFONATE, AND PROCESS FOR PRODUCTION OF CARBAMATE MITSUI CHEMICALS, INC. 2012-10-11 US disclosed
EP-2412703-A1 URETHANE COMPOUND AND PROCESS FOR PRODUCTION THEREOF, AND ISOCYANATE AND PROCESS FOR PRODUCTION THEREOF Mitsui Chemicals, Inc. (JP) 2012-02-01 EP disclosed
US-20120010427-A1 URETHANE COMPOUND AND METHOD FOR PRODUCING THE SAME, AND ISOCYANATE AND METHOD FOR PRODUCING THE SAME MITSUI CHEMICALS, INC. 2012-01-12 US disclosed