SCHEMBL4731272

SCHEMBL4731272

CC(C)c1ccc(Sc2cc(F)ccc2CC(=O)O)cc1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGBL2 Q5U5Z8 1/20 0.81
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 2/20 0.47
HPGD P15428 1/20 0.47
RXRA P19793 5/20 0.45
MMP2 P08253 1/20 0.41
MMP9 P14780 1/20 0.41
MMP12 P39900 1/20 0.41
PPARG P37231 1/20 0.40
PTGDR2 Q9Y5Y4 2/20 0.39
TBXA2R P21731 1/20 0.39
PTGDR Q13258 1/20 0.39
MEN1 O00255 1/20 0.39
CYP1A2 P05177 1/20 0.39
KMT2A Q03164 1/20 0.39
SLC6A9 P48067 3/20 0.39
RHEB Q15382 1/20 0.38
TSHR P16473 1/20 0.38
BCL2 P10415 1/20 0.37
MCL1 Q07820 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17296946 0.90 AGBL2 (1.00) AGBL2CYP2C9CYP2C19HPGDRXRA
SCHEMBL11407313 0.87 AGBL2 (0.62) AGBL2CYP2C9CYP2C19HPGDRXRA
SCHEMBL11343508 0.85 HPGD (0.65) AGBL2CYP2C9CYP2C19HPGDMMP2
SCHEMBL4733549 0.85 AGBL2 (0.59) AGBL2CYP2C9CYP2C19HPGDMMP2
SCHEMBL11335380 0.83 AGBL2 (0.56) AGBL2CYP2C9CYP2C19HPGDMMP2
SCHEMBL11338926 0.83 AGBL2 (0.56) AGBL2CYP2C9CYP2C19HPGDMMP2
SCHEMBL11334600 0.82 MMP2 (0.63) AGBL2CYP2C9CYP2C19HPGDMMP2
Fumaric Acid SCHEMBL8535167 0.80 AGBL2 (0.57) AGBL2RXRAKDM4E
Maleic Acid SCHEMBL8535164 0.80 AGBL2 (0.57) AGBL2RXRAKDM4E
SCHEMBL4732967 0.80 AGBL2 (0.62) AGBL2CYP2C9CYP2C19HPGDRXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008061029-A1 ARYL SULFONAMIDE DERIVATIVES AND METHODS OF THEIR USE WYETH (US) 2008-05-22 WO disclosed
US-4243805-A 3 Fluoro-10-piperazino-8-substituted 10,11-dihydrodibenzo-(bf) thiepins and method for the preparation thereof SPOFA, SPOJENE PODNIKY PRO ZDRAVOTNICKOU VYROBU (CS) 1981-01-06 US disclosed