SCHEMBL4731982

SCHEMBL4731982

FC(F)(F)c1cc(NC2CCN(c3ncccn3)CC2)ccc1Br

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SCD O00767 2/20 0.50
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
TRPV1 Q8NER1 2/20 0.41
DRD2 P14416 1/20 0.40
DRD3 P35462 1/20 0.40
CYP3A4 P08684 1/20 0.40
RBP4 P02753 1/20 0.39
MALT1 Q9UDY8 1/20 0.39
CCNC P24863 1/20 0.38
CDK8 P49336 1/20 0.38
MAPT P10636 2/20 0.38
RXFP1 Q9HBX9 1/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4733366 0.84 MALT1 (0.46) SCDSMN1; SMN2DRD2DRD3MALT1
SCHEMBL4729979 0.81 MALT1 (0.48) HTTSMN1; SMN2DRD2DRD3MALT1
SCHEMBL5096292 0.81 ALDH1A1 (0.47) HTTDRD2DRD3CYP3A4MAPT
SCHEMBL4731861 0.80 SCD (0.45) SCDHTTSMN1; SMN2TRPV1DRD2
SCHEMBL4728680 0.79 GRM4 (0.46) SMN1; SMN2DRD2DRD3MALT1MAPT
SCHEMBL4730521 0.79 SCD (0.58) SCDHTTSMN1; SMN2DRD2DRD3
SCHEMBL5094275 0.79 SLC6A7 (0.44) SCDMALT1CCNCCDK8MEN1
SCHEMBL4732425 0.78 FPR2 (0.49) SCDHTTSMN1; SMN2DRD2DRD3
SCHEMBL4733745 0.72 KDM4E (0.48) SMN1; SMN2MALT1
SCHEMBL5102640 0.70 MALT1 (0.49) SMN1; SMN2MALT1MAPTMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008058064-A1 AMINE-LINKED MULTICYCLIC COMPOUNDS AS INHIBITORS OF THE PROLINE TRANSPORTER LEXICON PHARMACEUTICALS, INC. (US) 2008-05-15 WO disclosed