SCHEMBL4733659

SCHEMBL4733659

CCN(CC)c1ccc(CN(C(=O)c2ccsc2)c2ccc(F)cc2)cn1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CACNA1H O95180 1/20 0.41
AOC3 Q16853 1/20 0.38
MAPK14 Q16539 1/20 0.38
LTB4R2 Q9NPC1 1/20 0.38
PDK1 Q15118 11/20 0.37
PDK2 Q15119 3/20 0.37
PDK3 Q15120 3/20 0.37
PDK4 Q16654 3/20 0.37
HSP90AA1 P07900 1/20 0.37
HSP90AB1 P08238 1/20 0.37
GRM1 Q13255 1/20 0.36
GRIA2 P42262 1/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2A Q12879 1/20 0.36
CXCR2 P25025 1/20 0.36
CNR2 P34972 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3821700 0.83 CNR2 (0.49) CACNA1HAOC3MAPK14LTB4R2PDK1
SCHEMBL4737075 0.83 MAPK14 (0.40) MAPK14LTB4R2PDK1PDK2PDK3
SCHEMBL4785417 0.82 CACNA1H (0.41) CACNA1HAOC3MAPK14LTB4R2PDK1
SCHEMBL4733787 0.82 KMT2A (0.48) CACNA1H
SCHEMBL4736030 0.81 CACNA1H (0.47) CACNA1HAOC3MAPK14LTB4R2CNR2
SCHEMBL3071006 0.81 CACNA1H (0.47) CACNA1HAOC3MAPK14LTB4R2GRIA2
Trifluoroacetic Acid SCHEMBL3825726 0.79 CNR2 (0.44) CACNA1HAOC3MAPK14LTB4R2PDK1
SCHEMBL3064331 0.78 CACNA1H (0.45) CACNA1HAOC3LTB4R2GRIA2GRIN1
SCHEMBL3815393 0.78 CACNA1H (0.45) CACNA1HAOC3LTB4R2GRIN1GRIN2A
SCHEMBL4734213 0.78 LMNA (0.54) CACNA1H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO claimed