SCHEMBL4734236

SCHEMBL4734236

CCC(C)(C)C(=O)Nc1cc(CN(C)S(=O)(=O)c2ccc(C(F)(F)F)cc2)c(Br)cn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 6/20 0.41
CNR1 P21554 4/20 0.41
KMT2A Q03164 2/20 0.40
NAMPT P43490 1/20 0.40
RAB9A P51151 1/20 0.38
TRPV4 Q9HBA0 1/20 0.38
AR P10275 1/20 0.38
ALDH1A1 P00352 2/20 0.38
RORC P51449 1/20 0.38
KDM4E B2RXH2 2/20 0.37
MEN1 O00255 1/20 0.37
MAPT P10636 1/20 0.37
BMP1 P13497 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MMP3 P08254 1/20 0.36
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
MMP1 P03956 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4730027 0.91 CNR2 (0.42) CNR2CNR1KMT2ANAMPTRAB9A
SCHEMBL4733445 0.78 RAB9A (0.40) CNR2CNR1KMT2ANAMPTRAB9A
SCHEMBL4733798 0.74 CNR2 (0.45) CNR2CNR1RAB9AALDH1A1KDM4E
SCHEMBL4731510 0.73 CNR2 (0.55) CNR2CNR1KMT2ARAB9AALDH1A1
SCHEMBL14206637 0.72 CNR2 (0.54) CNR2CNR1KMT2AALDH1A1MEN1
SCHEMBL14206962 0.72 CNR2 (0.45) CNR2CNR1KMT2AMEN1
SCHEMBL14206662 0.71 CNR2 (0.56) CNR2CNR1LMNA
SCHEMBL4734563 0.69 CNR2 (0.54) CNR2CNR1ARALDH1A1LMNA
SCHEMBL4733925 0.69 CNR2 (0.51) CNR2CNR1LMNA
SCHEMBL4731889 0.68 CNR2 (0.56) CNR2CNR1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008063625-A2 PYRIDINE COMPOUNDS AND METHODS OF THEIR USE ADOLOR CORPORATION (US) 2008-05-29 WO claimed
WO-2008063625-A2 PYRIDINE COMPOUNDS AND METHODS OF THEIR USE ADOLOR CORPORATION (US) 2008-05-29 WO disclosed