SCHEMBL4734328

SCHEMBL4734328

Cc1nc2c3c(c(C(N)=O)cc2n1C)CCC1(CCc2ccccc21)O3

nearest known ligand 0.32

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCNC P24863 3/20 0.32
CDK8 P49336 3/20 0.32
HASPIN Q8TF76 3/20 0.32
CDK19 Q9BWU1 3/20 0.32
ALDH1A1 P00352 1/20 0.32
TP53 P04637 1/20 0.32
PARP1 P09874 1/20 0.31
LDHA P00338 1/20 0.31
HRH1 P35367 2/20 0.31
PIN1 Q13526 3/20 0.30
BACE1 P56817 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4740444 0.91 HCAR2 (0.34) ALDH1A1TP53LDHAPIN1
SCHEMBL4735029 0.89 NPY5R (0.33) ALDH1A1TP53LDHA
SCHEMBL4784972 0.89 NPY5R (0.33) ALDH1A1TP53LDHA
SCHEMBL4737642 0.87 NPY5R (0.37) ALDH1A1
SCHEMBL4738064 0.87 AVPR1A (0.34) ALDH1A1
SCHEMBL4783797 0.86 RORC (0.38) ALDH1A1TP53
SCHEMBL4739249 0.86 PIN1 (0.31) PIN1
SCHEMBL4737057 0.85 OPRL1 (0.36) ALDH1A1
SCHEMBL4738895 0.84 KMT2A (0.36) ALDH1A1
SCHEMBL4737821 0.81 CYP26A1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008071765-A1 PHARMACEUTICALLY ACTIVE SPIRO-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES NYCOMED GMBH (DE) 2008-06-19 WO claimed
WO-2008071765-A1 PHARMACEUTICALLY ACTIVE SPIRO-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES NYCOMED GMBH (DE) 2008-06-19 WO disclosed