SCHEMBL4784972

SCHEMBL4784972

CNC(=O)c1cc2c(nc(C)n2C)c2c1CCC1(CCc3ccccc31)O2

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 1/20 0.33
SCN9A Q15858 1/20 0.32
NPC1 O15118 2/20 0.31
RAB9A P51151 2/20 0.31
TP53 P04637 2/20 0.31
ALDH1A1 P00352 1/20 0.31
LDHA P00338 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4740444 0.90 HCAR2 (0.34) TP53ALDH1A1LDHA
SCHEMBL4734328 0.89 CCNC (0.32) TP53ALDH1A1LDHA
SCHEMBL4737057 0.89 OPRL1 (0.36) RAB9AALDH1A1SMN1; SMN2
SCHEMBL4738895 0.87 KMT2A (0.36) NPC1RAB9AALDH1A1
SCHEMBL4735029 0.87 NPY5R (0.33) NPY5RTP53ALDH1A1LDHA
SCHEMBL4739802 0.87 NPC1 (0.32) NPC1RAB9ATP53SMN1; SMN2
SCHEMBL4737642 0.86 NPY5R (0.37) NPY5RNPC1RAB9AALDH1A1
SCHEMBL4738064 0.85 AVPR1A (0.34) ALDH1A1SMN1; SMN2
SCHEMBL4737821 0.85 CYP26A1 (0.39)
SCHEMBL4783797 0.84 RORC (0.38) TP53ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008071765-A1 PHARMACEUTICALLY ACTIVE SPIRO-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES NYCOMED GMBH (DE) 2008-06-19 WO claimed