SCHEMBL4734834

SCHEMBL4734834

COc1ccc(CN2C(=O)C(=O)c3cc(Br)c(Br)cc32)cc1

nearest known ligand 0.66

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.66
CA1 P00915 1/20 0.66
CA2 P00918 1/20 0.66
CA9 Q16790 1/20 0.66
PARK7 Q99497 1/20 0.65
CHRM5 P08912 5/20 0.62
CASP3 P42574 1/20 0.59
ACHE P22303 2/20 0.55
GSK3A P49840 1/20 0.54
GSK3B P49841 1/20 0.54
CMA1 P23946 1/20 0.53
TP53 P04637 1/20 0.51
MAPT P10636 1/20 0.51
ALDH1A1 P00352 1/20 0.49
ALDH2 P05091 1/20 0.49
ALDH3A1 P30838 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4782178 0.85 CHRM5 (0.68) CA12CA1CA2CA9PARK7
SCHEMBL4736417 0.82 PARK7 (0.73) CA12CA1CA2CA9PARK7
SCHEMBL3021031 0.80 CHRM5 (0.72) CA12CA1CA2CA9PARK7
SCHEMBL4738038 0.80 PARK7 (0.75) CA12CA1CA2CA9PARK7
SCHEMBL4735891 0.80 CHRM5 (0.68) CA12CA1CA2CA9PARK7
SCHEMBL18955136 0.80 CA1 (1.00) CA12CA1CA2CA9CHRM5
SCHEMBL4735921 0.79 PARK7 (1.00) CA12CA1CA2CA9PARK7
SCHEMBL29460856 0.79 CASP3 (0.76) CA12CA1CA2CA9CHRM5
SCHEMBL2305451 0.79 CASP3 (0.76) CA12CA1CA2CA9CHRM5
SCHEMBL4739205 0.77 CASP3 (0.54) CA12CA1CA2CA9PARK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008074078-A1 SELECTIVELY DELIVERABLE ISATIN-BASED CYTOTOXIC AGENTS UNIVERSITY OF WOLLONGONG (AU) 2008-06-26 WO disclosed