SCHEMBL4782178

SCHEMBL4782178

COc1ccc(CN2C(=O)C(=O)c3ccc(Br)cc32)cc1

nearest known ligand 0.68

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 5/20 0.68
PARK7 Q99497 1/20 0.64
ACHE P22303 2/20 0.60
CA12 O43570 1/20 0.58
CA1 P00915 1/20 0.58
CA2 P00918 1/20 0.58
CA9 Q16790 1/20 0.58
CASP3 P42574 1/20 0.58
CHRM1 P11229 1/20 0.57
CHRM3 P20309 1/20 0.57
ALDH1A1 P00352 2/20 0.54
ALDH3A1 P30838 2/20 0.54
ALDH2 P05091 1/20 0.54
GSK3A P49840 1/20 0.52
GSK3B P49841 1/20 0.52
CMA1 P23946 1/20 0.51
APAF1 O14727 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4734834 0.85 CA12 (0.66) CHRM5PARK7ACHECA12CA1
SCHEMBL28026703 0.83 ACHE (0.67) CHRM5ACHECA12CA1CA2
SCHEMBL31667682 0.82 CASP3 (0.62) CHRM5PARK7ACHECASP3GSK3A
SCHEMBL15206958 0.82 ALDH1A1 (0.78) CHRM5ACHECA12CA1CA2
SCHEMBL3014022 0.81 CHRM5 (0.67) CHRM5PARK7ACHECA12CA1
SCHEMBL2305451 0.81 CASP3 (0.76) CHRM5ACHECA12CA1CA2
SCHEMBL29460856 0.81 CASP3 (0.76) CHRM5ACHECA12CA1CA2
Nitrogen SCHEMBL28297413 0.80 ALDH1A1 (0.74) CHRM5ACHECA12CA1CA2
SCHEMBL7245333 0.79 ACHE (0.56) CHRM5PARK7ACHECA12CA1
SCHEMBL4735921 0.78 PARK7 (1.00) CHRM5PARK7CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008074078-A1 SELECTIVELY DELIVERABLE ISATIN-BASED CYTOTOXIC AGENTS UNIVERSITY OF WOLLONGONG (AU) 2008-06-26 WO disclosed