SCHEMBL4738147

SCHEMBL4738147

COc1ccc2c(c1)C(=CCc1c(C(=O)N(C)C)cc3c(nc(C)n3C)c1O)CC2

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 2/20 0.42
MTNR1A P48039 2/20 0.42
MTNR1B P49286 2/20 0.42
CYP19A1 P11511 5/20 0.36
CYP11B2 P19099 2/20 0.36
ACHE P22303 1/20 0.34
MAPT P10636 3/20 0.33
TP53 P04637 2/20 0.33
ABCB1 P08183 1/20 0.33
MAOB P27338 2/20 0.33
THRB P10828 1/20 0.32
RXFP1 Q9HBX9 1/20 0.31
MAOA P21397 2/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4739210 0.93 MIF (0.36) NQO2MTNR1AMTNR1BCYP19A1CYP11B2
SCHEMBL4735019 0.88 NQO2 (0.38) NQO2MTNR1AMTNR1BCYP19A1CYP11B2
SCHEMBL4737211 0.83 CYP19A1 (0.34) CYP19A1CYP11B2MAPTNPC1LMNA
SCHEMBL4737851 0.81 CYP19A1 (0.32) NQO2MTNR1AMTNR1BCYP19A1CYP11B2
SCHEMBL4734337 0.79 DUSP10 (0.31)
SCHEMBL4735621 0.77
SCHEMBL4736255 0.76 ALDH1A1 (0.39) MAPTALDH1A1RAB9ASMN1; SMN2
SCHEMBL4737338 0.74 KDM4E (0.36) NPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL4736286 0.74
SCHEMBL4735242 0.73 FNTA (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008071765-A1 PHARMACEUTICALLY ACTIVE SPIRO-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES NYCOMED GMBH (DE) 2008-06-19 WO disclosed