SCHEMBL4735211

SCHEMBL4735211

Cc1ccc(C(=O)N2CCC(c3ccccc3)CC2)cc1N

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.58
CA1 P00915 1/20 0.58
CA2 P00918 1/20 0.58
CA7 P43166 1/20 0.58
CA9 Q16790 1/20 0.58
CA14 Q9ULX7 1/20 0.58
PARP14 Q460N5 2/20 0.56
PARP10 Q53GL7 2/20 0.56
HSD11B1 P28845 3/20 0.55
ALDH1A1 P00352 4/20 0.52
TP53 P04637 2/20 0.52
HPGD P15428 1/20 0.52
NPC1 O15118 2/20 0.51
RAB9A P51151 2/20 0.51
ATM Q13315 1/20 0.51
KDM4E B2RXH2 2/20 0.50
LMNA P02545 2/20 0.49
TSHR P16473 1/20 0.49
TRPV6 Q9H1D0 1/20 0.48
MAPT P10636 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14209216 0.90 ALDH1A1 (0.52) CA12CA1CA2CA7CA9
SCHEMBL4733674 0.90 ALDH1A1 (0.52) ALDH1A1TP53HPGDLMNAMAPT
SCHEMBL4175647 0.89 PARP10 (0.56) PARP14PARP10ALDH1A1TP53HPGD
SCHEMBL4197739 0.88 FASN (0.61) ALDH1A1TP53HPGDMAPTFASN
SCHEMBL16799271 0.88 HPGD (0.50) ALDH1A1TP53HPGDLMNATSHR
SCHEMBL4191753 0.88 PARP10 (0.58) PARP14PARP10HSD11B1ALDH1A1TP53
SCHEMBL4731334 0.85 FASN (0.63) PARP14PARP10HSD11B1ALDH1A1HPGD
SCHEMBL4735697 0.85 LMNA (0.51) PARP10HSD11B1ALDH1A1TP53HPGD
SCHEMBL4195205 0.85 ALDH1A1 (0.48) ALDH1A1TP53HPGDLMNAFASN
SCHEMBL14210109 0.85 KDM4E (0.47) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008059214-A1 BISAMLDE DERIVATIVES AND USE THEREOF AS FATTY ACID SYNTHASE INHIBITORS ASTRAZENECA AB (SE) 2008-05-22 WO disclosed