SCHEMBL4735626

SCHEMBL4735626

O=C(c1cccnc1)N(Cc1ccc(N2CCN(CCC3CCCCC3)CC2)nc1)c1ccc(F)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.42
GAA P10253 1/20 0.42
HTR2A P28223 6/20 0.41
DRD3 P35462 6/20 0.41
HTR1A P08908 5/20 0.41
DRD4 P21917 4/20 0.41
HTR7 P34969 4/20 0.41
DRD2 P14416 6/20 0.40
OPRM1 P35372 1/20 0.40
OPRK1 P41145 1/20 0.40
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
HTR2C P28335 2/20 0.38
TMEM97 Q5BJF2 2/20 0.38
SIGMAR1 Q99720 2/20 0.38
SMO Q99835 1/20 0.38
HSD17B10 Q99714 1/20 0.38
SLC6A4 P31645 1/20 0.38
PDK1 Q15118 1/20 0.38
SLC6A9 P48067 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4736483 0.88 TSHR (0.47) TSHRGAAHTR2ADRD3HTR1A
SCHEMBL4733572 0.87 TSHR (0.45) TSHRGAAOPRM1OPRK1ALDH1A1
SCHEMBL4735150 0.87 TSHR (0.51) TSHRGAAOPRM1OPRK1ALDH1A1
SCHEMBL4738289 0.86 GAA (0.45) TSHRGAAOPRM1KDM4ESMO
SCHEMBL4737126 0.86 TSHR (0.48) TSHRGAAHTR2ADRD3HTR1A
SCHEMBL4735433 0.86 OPRM1 (0.40) TSHRHTR2ADRD3HTR1ADRD4
SCHEMBL4785409 0.85 TSHR (0.52) TSHRGAAHTR2ADRD3HTR1A
SCHEMBL4738239 0.85 TSHR (0.49) TSHRGAAHTR2ADRD3HTR1A
SCHEMBL4737945 0.85 OPRM1 (0.44) TSHRHTR2ADRD3HTR1ADRD4
SCHEMBL4735235 0.84 GAA (0.47) TSHRGAAOPRM1KDM4ESMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO claimed
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO disclosed