SCHEMBL473596

SCHEMBL473596

O=C(O)c1cnccc1-c1cccc(C(F)(F)F)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 2/20 0.53
RORC P51449 1/20 0.50
RORB Q92753 1/20 0.50
KLRK1 P26718 1/20 0.48
MICA Q29983 1/20 0.48
RAET1L Q5VY80 1/20 0.48
EPHX2 P34913 1/20 0.47
DHODH Q02127 3/20 0.47
GPBAR1 Q8TDU6 1/20 0.46
ALDH1A1 P00352 3/20 0.45
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
KDM4E B2RXH2 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
XDH P47989 1/20 0.45
PIN1 Q13526 1/20 0.45
GMNN O75496 1/20 0.45
LMNA P02545 1/20 0.45
TTR P02766 1/20 0.45
CYP1A2 P05177 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1398852 0.81 RORB (0.68) KMORORCRORBALDH1A1MEN1
SCHEMBL4246561 0.80 DHODH (0.55) KMODHODHALDH1A1MEN1KMT2A
SCHEMBL34469496 0.80 PARP1 (0.54) KMORORCRORBKLRK1MICA
SCHEMBL5851623 0.79 RORC (0.54) KMORORCRORBALDH1A1KDM4E
SCHEMBL2222831 0.78 ALDH1A1 (0.50) DHODHALDH1A1MEN1KMT2AKDM4E
SCHEMBL7423738 0.78 RPS6KA3 (0.53) KMODHODHALDH1A1MEN1KMT2A
SCHEMBL22489951 0.78 MEN1 (0.44) KLRK1MICARAET1LDHODHGPBAR1
SCHEMBL10364611 0.77 MKNK1 (0.56) KMODHODHALDH1A1MEN1KMT2A
SCHEMBL30705023 0.77 MKNK1 (0.56) KMODHODHALDH1A1MEN1KMT2A
Hydrochloric Acid SCHEMBL7279409 0.77 ALDH1A1 (0.49) DHODHALDH1A1MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411011-A1 NOVEL AMINOPYRIDINE DERIVATIVES HAVING AURORA A SELECTIVE INHIBITORY ACTION MSD K.K. (JP) 2012-02-01 EP disclosed
WO-2010111056-A1 NOVEL AMINOPYRIDINE DERIVATIVES HAVING AURORA A SELECTIVE INHIBITORY ACTION BANYU PHARMACEUTICAL CO., LTD. (JP) 2010-09-30 WO disclosed