SCHEMBL7423738

SCHEMBL7423738

Cc1cccc(-c2ccncc2C(=O)O)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RPS6KA3 P51812 1/20 0.53
KMO O15229 2/20 0.50
KDM4E B2RXH2 2/20 0.48
LMNA P02545 1/20 0.48
HTT P42858 1/20 0.48
AKR1C2 P52895 1/20 0.47
AKR1C1 Q04828 1/20 0.47
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
DHODH Q02127 4/20 0.44
LDHA P00338 1/20 0.44
CDC7 O00311 1/20 0.44
KDM4C Q9H3R0 2/20 0.43
KDM6B O15054 1/20 0.43
CNR2 P34972 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HSD17B10 Q99714 1/20 0.43
DDT P30046 1/20 0.43
PIN1 Q13526 1/20 0.43
CYP2A6 P11509 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2560779 0.82 DDT (0.51) RPS6KA3KMOKDM4ELMNAHTT
SCHEMBL2222831 0.82 ALDH1A1 (0.50) RPS6KA3KDM4EHTTMEN1KMT2A
SCHEMBL10364611 0.80 MKNK1 (0.56) KMOKDM4ELMNAHTTMEN1
Hydrochloric Acid SCHEMBL7279409 0.80 ALDH1A1 (0.49) RPS6KA3KDM4EHTTMEN1KMT2A
SCHEMBL30705023 0.80 MKNK1 (0.56) KMOKDM4ELMNAHTTMEN1
SCHEMBL2557801 0.79 TRIM24 (0.50) KMOKDM4ELMNAHTTMEN1
SCHEMBL30361685 0.79 L3MBTL1 (0.59) KMOKDM4EAKR1C2AKR1C1MEN1
SCHEMBL268963 0.79 L3MBTL1 (0.59) KMOKDM4EAKR1C2AKR1C1MEN1
SCHEMBL473596 0.78 KMO (0.53) KMOKDM4ELMNAAKR1C2MEN1
SCHEMBL4248571 0.78 KDM4E (0.60) KMOKDM4ELMNAHTTAKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1263755-A2 CYCLIC BETA-AMINO ACID DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEASES AND TNF-ALPHA Bristol-Myers Squibb Pharma Company (US) 2002-12-11 EP disclosed
WO-2001070673-A2 CYCLIC β-AMINO ACID DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEASES AND TNF-$g(a) BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2001-09-27 WO disclosed