SCHEMBL4736076

SCHEMBL4736076

COc1c(CC=O)cc(C(C)(C)C)cc1C(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RXRA P19793 9/20 0.40
PPARG P37231 8/20 0.40
RARG P13631 4/20 0.40
ALDH1A1 P00352 1/20 0.36
TSHR P16473 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
TNFRSF1A P19438 2/20 0.35
DHFR P00374 1/20 0.34
PTGS2 P35354 2/20 0.33
PTGS1 P23219 1/20 0.33
HTR2A P28223 1/20 0.32
CYP2C19 P33261 1/20 0.32
RARA P10276 1/20 0.32
RARB P10826 1/20 0.32
RXRB P28702 1/20 0.32
RXRG P48443 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13368066 0.84 RXRA (0.40) RXRAPPARGRARGALDH1A1TSHR
SCHEMBL4734116 0.84 RXRA (0.47) RXRAPPARGRARGALDH1A1TSHR
SCHEMBL4731223 0.81 CYP2C19 (0.30) CYP2C19
SCHEMBL7921794 0.80 RXRA (0.50) RXRAPPARGRARGRARARARB
SCHEMBL6407060 0.79 MAPT (0.42) RXRAPPARGRARGALDH1A1TSHR
SCHEMBL15590742 0.79 RXRA (0.36) RXRAPPARGRARGALDH1A1TSHR
SCHEMBL4730685 0.79 DHFR (0.43) RXRAPPARGRARGALDH1A1TSHR
SCHEMBL4729047 0.78 ALDH1A1 (0.45) ALDH1A1TSHRPTGS2CYP2C19
SCHEMBL2947022 0.78 PTGS2 (0.47) RXRAPPARGRARGALDH1A1TSHR
SCHEMBL7796138 0.78 RXRA (0.44) RXRAPPARGRARGALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008052288-A1 DITHIOLE COMPOUNDS AS COX INHIBITORS NEURO THERAPEUTICS LIMITED (AU) 2008-05-08 WO disclosed