SCHEMBL4736255

SCHEMBL4736255

CCOC(=O)c1cc2c(nc(C)n2C)c(O)c1CC=C1CCc2ccccc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.39
KDM4E B2RXH2 5/20 0.39
HPGD P15428 4/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
KMT2A Q03164 2/20 0.36
HSP90AA1 P07900 2/20 0.36
POLB P06746 2/20 0.36
MAPT P10636 2/20 0.36
MEN1 O00255 1/20 0.36
USP2 O75604 1/20 0.36
TSHR P16473 1/20 0.36
RAB9A P51151 1/20 0.36
HSP90AB1 P08238 1/20 0.35
HSD17B10 Q99714 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
GABRG2 P18507 3/20 0.34
GABRB3 P28472 3/20 0.34
GABRA5 P31644 3/20 0.34
GABRP O00591 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4739791 0.89 TSHR (0.36) ALDH1A1KDM4EHPGDKMT2AMEN1
SCHEMBL4737293 0.88 ALDH1A1 (0.37) ALDH1A1KDM4EHPGDTDP1L3MBTL1
SCHEMBL4737295 0.88 ALDH1A1 (0.37) ALDH1A1KDM4EHPGDTDP1L3MBTL1
SCHEMBL4737617 0.78 TSHR (0.33) ALDH1A1KMT2AMEN1TSHRSMN1; SMN2
SCHEMBL4738147 0.76 NQO2 (0.42) ALDH1A1MAPTRAB9ASMN1; SMN2
SCHEMBL4736257 0.76 ALDH1A1 (0.32) ALDH1A1KDM4EL3MBTL1KMT2AMAPT
SCHEMBL4664575 0.74 KMT2A (0.41) ALDH1A1KDM4EHPGDKMT2AMAPT
SCHEMBL4737211 0.74 CYP19A1 (0.34) KMT2APOLBMAPTMEN1RAB9A
SCHEMBL5116642 0.73 GAA (0.43) ALDH1A1KDM4EHPGDL3MBTL1KMT2A
SCHEMBL4735946 0.73 ELANE (0.40) ALDH1A1KDM4EHPGDL3MBTL1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008071765-A1 PHARMACEUTICALLY ACTIVE SPIRO-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES NYCOMED GMBH (DE) 2008-06-19 WO disclosed