SCHEMBL4737211

SCHEMBL4737211

COc1cccc2c1C(=CCc1c(C(=O)N(C)C)cc3c(nc(C)n3C)c1O)CC2

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
PTK2 Q05397 1/20 0.32
NPC1 O15118 3/20 0.31
MAPT P10636 3/20 0.31
RAB9A P51151 3/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
HRH3 Q9Y5N1 2/20 0.31
F2 P00734 1/20 0.31
F10 P00742 1/20 0.31
TUBB4A P04350 1/20 0.31
TUBB P07437 1/20 0.31
TUBA3C P0DPH7 1/20 0.31
TUBA1B P68363 1/20 0.31
TUBA4A P68366 1/20 0.31
TUBB4B P68371 1/20 0.31
TUBB3 Q13509 1/20 0.31
TUBB2A Q13885 1/20 0.31
TUBB8 Q3ZCM7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4739807 0.89 PTK2 (0.31) CYP19A1CYP11B1CYP11B2PTK2
SCHEMBL4738147 0.83 NQO2 (0.42) CYP19A1CYP11B2NPC1MAPTRAB9A
SCHEMBL4739210 0.83 MIF (0.36) CYP19A1CYP11B1CYP11B2NPC1MAPT
SCHEMBL4964361 0.75 IDO1 (0.38) NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL4736255 0.74 ALDH1A1 (0.39) MAPTRAB9ASMN1; SMN2MEN1POLB
SCHEMBL4737338 0.73 KDM4E (0.36) NPC1RAB9ASMN1; SMN2MEN1GAA
SCHEMBL4735019 0.73 NQO2 (0.38) CYP19A1CYP11B2MAPT
SCHEMBL4737851 0.73 CYP19A1 (0.32) CYP19A1CYP11B1CYP11B2NPC1MAPT
SCHEMBL4735017 0.72
SCHEMBL4735621 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008071765-A1 PHARMACEUTICALLY ACTIVE SPIRO-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES NYCOMED GMBH (DE) 2008-06-19 WO disclosed