SCHEMBL4736285

SCHEMBL4736285

COCCCn1nc(C)c2ccc(C#CCO)cc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
REN P00797 5/20 0.44
KMO O15229 1/20 0.39
HRH3 Q9Y5N1 1/20 0.37
ADORA2A P29274 2/20 0.36
ADORA2B P29275 2/20 0.36
GLS O94925 1/20 0.34
SLC22A12 Q96S37 7/20 0.33
MELK Q14680 1/20 0.33
NR3C1 P04150 1/20 0.32
TUBB4A P04350 1/20 0.32
TUBB P07437 1/20 0.32
TUBA3C P0DPH7 1/20 0.32
TUBA1B P68363 1/20 0.32
TUBA4A P68366 1/20 0.32
TUBB4B P68371 1/20 0.32
TUBB3 Q13509 1/20 0.32
TUBB2A Q13885 1/20 0.32
TUBB8 Q3ZCM7 1/20 0.32
TUBA3E Q6PEY2 1/20 0.32
TUBA1A Q71U36 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13132264 0.79 REN (0.46) RENKMOADORA2AADORA2BGLS
SCHEMBL91359 0.79 REN (0.46) RENKMOADORA2AADORA2BGLS
SCHEMBL4732483 0.78 REN (0.40) RENHRH3SLC22A12
SCHEMBL1051150 0.76 REN (0.45) RENKMOADORA2AADORA2BGLS
SCHEMBL4249553 0.76 REN (0.45) RENKMOADORA2AADORA2BGLS
SCHEMBL13448565 0.76 REN (0.45) RENKMOADORA2AADORA2BGLS
SCHEMBL13131423 0.75 ADORA2A (0.44) RENKMOADORA2AADORA2BGLS
SCHEMBL78153 0.74 REN (0.55) RENKMOADORA2AADORA2BGLS
SCHEMBL4253933 0.74 REN (0.45) RENKMOADORA2AADORA2BGLS
SCHEMBL2807350 0.74 REN (0.48) RENKMOSLC22A12NR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008055939-A2 PROCESS FOR PREPARING 2-ALKYL-3-HETEROCYCLYL- PROP-2-EN- 1-OL DERIVATIVES NOVARTIS AG (CH) 2008-05-15 WO disclosed