SCHEMBL91359

SCHEMBL91359

COCCCn1nc(C)c2ccc(C)cc21

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
REN P00797 6/20 0.46
ADORA2A P29274 2/20 0.44
ADORA2B P29275 2/20 0.44
KMO O15229 1/20 0.43
GLS O94925 1/20 0.41
PDE5A O76074 1/20 0.37
SCN9A Q15858 1/20 0.37
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
SLC22A12 Q96S37 3/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
NR3C1 P04150 1/20 0.35
ALDH1A1 P00352 1/20 0.35
ESR1 P03372 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1051150 0.86 REN (0.45) RENADORA2AADORA2BKMOGLS
SCHEMBL13131423 0.85 ADORA2A (0.44) RENADORA2AADORA2BKMOGLS
SCHEMBL13132264 0.83 REN (0.46) RENADORA2AADORA2BKMOGLS
SCHEMBL78153 0.83 REN (0.55) RENADORA2AADORA2BKMOGLS
SCHEMBL4249553 0.82 REN (0.45) RENADORA2AADORA2BKMOGLS
SCHEMBL13448565 0.82 REN (0.45) RENADORA2AADORA2BKMOGLS
SCHEMBL4256101 0.82 GLS (0.62) RENGLSMEN1KMT2AALDH1A1
SCHEMBL2807350 0.80 REN (0.48) RENKMOHTTSLC22A12KMT2A
SCHEMBL14752740 0.79 ADORA2A (0.44) ADORA2AADORA2BKMOGLSSLC22A12
SCHEMBL4736285 0.79 REN (0.44) RENADORA2AADORA2BKMOGLS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed