SCHEMBL4736729

SCHEMBL4736729

CN1CCCN(c2ccc(CN(C(=O)c3cccnc3)c3ccc(F)cc3)cn2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.46
GAA P10253 1/20 0.46
PDK1 Q15118 5/20 0.44
OPRM1 P35372 2/20 0.43
OPRK1 P41145 1/20 0.43
CXCR2 P25025 1/20 0.40
HTT P42858 1/20 0.40
HTR1A P08908 2/20 0.39
DRD2 P14416 2/20 0.39
DRD4 P21917 2/20 0.39
HTR2A P28223 2/20 0.39
HTR2C P28335 2/20 0.39
HTR7 P34969 2/20 0.39
DRD3 P35462 2/20 0.39
TMEM97 Q5BJF2 2/20 0.39
SIGMAR1 Q99720 2/20 0.39
SLC6A4 P31645 1/20 0.39
MAPK14 Q16539 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39
KCNH2 Q12809 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4738239 0.96 TSHR (0.49) TSHRGAAPDK1OPRM1OPRK1
SCHEMBL4735150 0.91 TSHR (0.51) TSHRGAAPDK1OPRM1OPRK1
SCHEMBL4737126 0.89 TSHR (0.48) TSHRGAAPDK1OPRM1OPRK1
SCHEMBL4736584 0.88 TSHR (0.51) TSHRGAAPDK1OPRM1OPRK1
SCHEMBL4739086 0.88 TSHR (0.52) TSHRGAAPDK1CXCR2HTT
SCHEMBL3830332 0.87 MEN1 (0.45) TSHRGAAOPRM1OPRK1CXCR2
SCHEMBL4736483 0.87 TSHR (0.47) TSHRGAAPDK1OPRM1OPRK1
SCHEMBL8185382 0.87 RAB9A (0.48) PDK1OPRM1OPRK1HTR1ADRD2
SCHEMBL4735615 0.86 MAPK14 (0.45) TSHROPRM1OPRK1CXCR2HTR1A
SCHEMBL4736473 0.86 OPRM1 (0.41) TSHROPRM1OPRK1CXCR2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO claimed