SCHEMBL4737404

SCHEMBL4737404

COc1cccc(CN2C(=O)C(=O)c3cc(Br)cc(Br)c32)c1

nearest known ligand 0.76

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PARK7 Q99497 5/20 0.76
CHRM5 P08912 4/20 0.58
CMA1 P23946 1/20 0.56
ALDH1A1 P00352 6/20 0.52
ALDH3A1 P30838 5/20 0.52
ALDH2 P05091 4/20 0.52
MAPT P10636 3/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
KDM4E B2RXH2 1/20 0.51
MEN1 O00255 1/20 0.51
POLB P06746 1/20 0.51
HPGD P15428 1/20 0.51
MAPK1 P28482 1/20 0.51
KMT2A Q03164 1/20 0.51
ATM Q13315 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
TP53 P04637 2/20 0.50
TDP1 Q9NUW8 1/20 0.48
GAA P10253 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4785342 0.89 PARK7 (0.72) PARK7CHRM5CMA1ALDH1A1ALDH3A1
SCHEMBL4735921 0.86 PARK7 (1.00) PARK7CHRM5CMA1ALDH1A1ALDH3A1
SCHEMBL4736331 0.82 PARK7 (0.75) PARK7CHRM5ALDH1A1ALDH3A1ALDH2
SCHEMBL4784997 0.80 PARK7 (0.57) PARK7ALDH1A1MAPTSMN1; SMN2KDM4E
SCHEMBL4786048 0.80 PARK7 (0.78) PARK7CHRM5ALDH1A1ALDH3A1ALDH2
SCHEMBL4784829 0.79 PARK7 (0.67) PARK7CHRM5ALDH1A1ALDH3A1ALDH2
SCHEMBL12930258 0.79 CHRM5 (0.81) PARK7CHRM5CMA1ALDH1A1ALDH3A1
SCHEMBL12930254 0.79 CHRM5 (0.61) PARK7CHRM5CMA1ALDH1A1ALDH3A1
SCHEMBL30774299 0.78 PARK7 (0.82) PARK7CHRM5ALDH1A1ALDH3A1ALDH2
SCHEMBL4739092 0.78 PARK7 (0.82) PARK7CHRM5ALDH1A1ALDH3A1ALDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008074078-A1 SELECTIVELY DELIVERABLE ISATIN-BASED CYTOTOXIC AGENTS UNIVERSITY OF WOLLONGONG (AU) 2008-06-26 WO disclosed