SCHEMBL4737745

SCHEMBL4737745

N[C@](CO)(C(=O)O)[C@@H](O)CCCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 1/20 0.47
TRPA1 O75762 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.43
HDAC3 O15379 2/20 0.43
HDAC4 P56524 2/20 0.43
HDAC1 Q13547 2/20 0.43
HDAC7 Q8WUI4 2/20 0.43
HDAC2 Q92769 2/20 0.43
HDAC10 Q969S8 2/20 0.43
HDAC11 Q96DB2 2/20 0.43
HDAC8 Q9BY41 2/20 0.43
HDAC6 Q9UBN7 2/20 0.43
HDAC9 Q9UKV0 2/20 0.43
HDAC5 Q9UQL6 2/20 0.43
MAPK1 P28482 1/20 0.43
ADRA1A P35348 1/20 0.43
SLC6A3 Q01959 1/20 0.43
GRM2 Q14416 2/20 0.43
GRM3 Q14832 2/20 0.43
HIF1A Q16665 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14145254 1.00 GRIK1 (0.47) GRIK1TRPA1SMN1; SMN2HDAC3HDAC4
SCHEMBL14145666 0.90 GRIK1 (0.43) GRIK1TRPA1SMN1; SMN2HDAC3HDAC4
SCHEMBL14145246 0.88 GRIK1 (0.44) GRIK1TRPA1SMN1; SMN2HDAC3HDAC4
SCHEMBL14201435 0.84 TRPA1 (0.49) GRIK1TRPA1SMN1; SMN2HDAC3HDAC4
SCHEMBL13953256 0.83 ALOX5 (0.48) TDP1PPARAALOX5
SCHEMBL14201498 0.81 GRIK1 (0.50) GRIK1TRPA1SMN1; SMN2HDAC3HDAC4
SCHEMBL14201434 0.81 GRIK1 (0.50) GRIK1TRPA1SMN1; SMN2HDAC3HDAC4
SCHEMBL14145649 0.80 ALDH1A1 (0.42) TRPA1SMN1; SMN2MMP2
SCHEMBL14259474 0.78 GRIK1 (0.49) GRIK1TRPA1MMP2MMP3
SCHEMBL14201480 0.78 SMN1; SMN2 (0.42) TRPA1SMN1; SMN2GRM2GRM3HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008083280-A1 COMPOUNDS AND METHODS OF TREATING INSULIN RESISTANCE AND CARDIOMYOPATHY TRANSITION THERAPEUTICS INC. (CA) 2008-07-10 WO disclosed