SCHEMBL4739340

SCHEMBL4739340

O=C(CC(NC(=O)c1cnc2cc(F)ccc2c1N1CCNCC1)C(=O)CF)OC(=O)C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.40
CASP3 P42574 1/20 0.35
ALDH1A1 P00352 7/20 0.33
HDAC3 O15379 5/20 0.33
HDAC2 Q92769 1/20 0.33
CCNC P24863 1/20 0.33
CDK8 P49336 1/20 0.33
ADRB2 P07550 1/20 0.33
NCF1 P14598 1/20 0.33
WDR5 P61964 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4742120 0.92 THRB (0.43) THRBCASP3ADRB2NCF1
SCHEMBL4742118 0.89 MET (0.38) THRBALDH1A1
SCHEMBL4743039 0.85 USP2 (0.35) CASP3ALDH1A1
SCHEMBL4739980 0.84 THRB (0.44) THRBCASP3ALDH1A1CCNCCDK8
Trifluoroacetic Acid SCHEMBL4742140 0.74 THRB (0.43) THRBCASP3ALDH1A1
SCHEMBL4785468 0.74 THRB (0.45) THRB
Trifluoroacetic Acid SCHEMBL4785493 0.72 THRB (0.45) THRBCASP3ALDH1A1
SCHEMBL4743062 0.72 THRB (0.47) THRBCASP3ALDH1A1
SCHEMBL4739351 0.72 MAPK1 (0.35) ALDH1A1WDR5
SCHEMBL4741648 0.71 THRB (0.43) THRBCASP3ALDH1A1CCNCCDK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008093940-A1 QUINOLINE DERIVATIVES AS CASPASE-3 INHIBITOR, PREPARATION PROCESS FOR THE SAME AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME YUNGJIN PHARMACEUTICAL CO., LTD. (KR) 2008-08-07 WO claimed
WO-2008093940-A1 QUINOLINE DERIVATIVES AS CASPASE-3 INHIBITOR, PREPARATION PROCESS FOR THE SAME AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME YUNGJIN PHARMACEUTICAL CO., LTD. (KR) 2008-08-07 WO disclosed