SCHEMBL4743039

SCHEMBL4743039

O=C(CC(NC(=O)c1cnc2c(F)cccc2c1N1CCNCC1)C(=O)CF)OC(=O)C(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.35
TP53 P04637 1/20 0.35
MAPK1 P28482 1/20 0.35
RECQL P46063 1/20 0.35
HSD17B10 Q99714 1/20 0.35
MAPT P10636 3/20 0.35
SCN9A Q15858 1/20 0.31
TACR3 P29371 1/20 0.31
KCNH2 Q12809 1/20 0.31
CASP3 P42574 3/20 0.31
KDM4E B2RXH2 2/20 0.31
LMNA P02545 2/20 0.31
NPSR1 Q6W5P4 2/20 0.31
GLA P06280 1/20 0.31
HTT P42858 1/20 0.31
NTRK1 P04629 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
KMT2A Q03164 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4742554 0.92 TP53 (0.36) USP2TP53MAPK1RECQLHSD17B10
SCHEMBL4742130 0.92 USP2 (0.45) USP2TP53MAPK1RECQLHSD17B10
SCHEMBL4742618 0.90 USP2 (0.34) USP2TP53MAPK1RECQLHSD17B10
SCHEMBL4739340 0.85 THRB (0.40) CASP3ALDH1A1
SCHEMBL4742120 0.83 THRB (0.43) SCN9AKCNH2CASP3
SCHEMBL4739351 0.81 MAPK1 (0.35) USP2TP53MAPK1RECQLHSD17B10
SCHEMBL4742118 0.80 MET (0.38) RECQLMAPTKDM4ELMNANPSR1
SCHEMBL4742574 0.78 DRD2 (0.35) USP2TP53MAPK1RECQLHSD17B10
SCHEMBL4739980 0.75 THRB (0.44) MAPTCASP3ALDH1A1SMN1; SMN2
SCHEMBL4742621 0.72 USP2 (0.45) USP2TP53MAPK1RECQLHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008093940-A1 QUINOLINE DERIVATIVES AS CASPASE-3 INHIBITOR, PREPARATION PROCESS FOR THE SAME AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME YUNGJIN PHARMACEUTICAL CO., LTD. (KR) 2008-08-07 WO claimed
WO-2008093940-A1 QUINOLINE DERIVATIVES AS CASPASE-3 INHIBITOR, PREPARATION PROCESS FOR THE SAME AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME YUNGJIN PHARMACEUTICAL CO., LTD. (KR) 2008-08-07 WO disclosed