SCHEMBL473989

SCHEMBL473989

CC(c1cccc(-c2ccccc2)c1C(=O)O)C(O)(c1ccc2c(c1)N(C)C(=O)CO2)C(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
NR1H2 P55055 2/20 0.34
NR1H3 Q13133 2/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
GPR55 Q9Y2T6 1/20 0.34
CMA1 P23946 1/20 0.34
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
THRB P10828 1/20 0.34
PTGER3 P43115 1/20 0.34
MALT1 Q9UDY8 1/20 0.34
ALOX12 P18054 1/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
TP53 P04637 2/20 0.33
MAPT P10636 1/20 0.33
KDM4E B2RXH2 1/20 0.33
POLB P06746 1/20 0.33
HTR1A P08908 1/20 0.32
HTR2C P28335 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL473958 0.86 ALDH1A1 (0.37) ALDH1A1NR1H2NR1H3L3MBTL1GPR55
SCHEMBL473903 0.86 ALDH1A1 (0.37) ALDH1A1NR1H2NR1H3L3MBTL1GPR55
SCHEMBL474394 0.82 POLB (0.36) ALDH1A1L3MBTL1GPR55PDE3BPDE3A
SCHEMBL474579 0.81 GPR55 (0.35) ALDH1A1NR1H2NR1H3L3MBTL1GPR55
SCHEMBL12163813 0.81 GPR55 (0.35) ALDH1A1NR1H2NR1H3L3MBTL1GPR55
SCHEMBL12163808 0.80 GPR55 (0.37) ALDH1A1GPR55PDE3BPDE3ATHRB
SCHEMBL474290 0.80 GPR55 (0.37) ALDH1A1GPR55PDE3BPDE3ATHRB
SCHEMBL12163784 0.80 GPR55 (0.37) ALDH1A1GPR55PDE3BPDE3ATHRB
SCHEMBL474474 0.80 GPR55 (0.37) ALDH1A1GPR55PDE3BPDE3ATHRB
SCHEMBL474495 0.79 BDKRB1 (0.42) GPR55

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed