SCHEMBL473903

SCHEMBL473903

CC(c1c(C(=O)O)cccc1-c1ccccc1)C(O)(c1ccc2c(c1)N(C)C(=O)CO2)C(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 1/20 0.36
NR1H2 P55055 2/20 0.36
NR1H3 Q13133 2/20 0.36
CMA1 P23946 1/20 0.36
MALT1 Q9UDY8 1/20 0.35
GPR55 Q9Y2T6 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
THRB P10828 1/20 0.34
PTGER3 P43115 1/20 0.34
MAP3K5 Q99683 1/20 0.33
ALOX12 P18054 1/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
MAPT P10636 2/20 0.33
TP53 P04637 1/20 0.33
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL473989 0.86 ALDH1A1 (0.37) ALDH1A1KDM4ENR1H2NR1H3CMA1
SCHEMBL473958 0.83 ALDH1A1 (0.37) ALDH1A1KDM4ENR1H2NR1H3MALT1
SCHEMBL12163813 0.83 GPR55 (0.35) ALDH1A1KDM4ENR1H2NR1H3CMA1
SCHEMBL474579 0.83 GPR55 (0.35) ALDH1A1KDM4ENR1H2NR1H3CMA1
SCHEMBL474394 0.78 POLB (0.36) ALDH1A1MALT1GPR55L3MBTL1PDE3B
SCHEMBL474521 0.78 TP53 (0.39) ALDH1A1NR1H3CMA1TP53
SCHEMBL473961 0.78 ALDH1A1 (0.41) ALDH1A1CMA1THRBCYP11B2MAPT
SCHEMBL474057 0.77 KMO (0.36) ALDH1A1NR1H2NR1H3CMA1THRB
SCHEMBL474348 0.77 GPR55 (0.39) ALDH1A1CMA1MALT1GPR55L3MBTL1
SCHEMBL12163826 0.77 GPR55 (0.39) ALDH1A1CMA1MALT1GPR55L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed