SCHEMBL473958

SCHEMBL473958

CC(c1cc(C(=O)O)ccc1-c1ccccc1)C(O)(c1ccc2c(c1)N(C)C(=O)CO2)C(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
PTGER3 P43115 1/20 0.35
USP30 Q70CQ3 1/20 0.35
GPR55 Q9Y2T6 1/20 0.34
LMNA P02545 1/20 0.34
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
MGLL Q99685 1/20 0.33
KDM4E B2RXH2 1/20 0.33
POLB P06746 1/20 0.33
NR1H2 P55055 1/20 0.32
NR1H3 Q13133 1/20 0.32
MALT1 Q9UDY8 1/20 0.32
TBXA2R P21731 2/20 0.32
RIPK1 Q13546 1/20 0.32
THRB P10828 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL474394 0.92 POLB (0.36) ALDH1A1L3MBTL1PTGER3USP30GPR55
SCHEMBL474455 0.87 ALDH1A1 (0.34) ALDH1A1LMNAMALT1
SCHEMBL474284 0.87 ALDH1A1 (0.38) ALDH1A1L3MBTL1PTGER3USP30GPR55
SCHEMBL473989 0.86 ALDH1A1 (0.37) ALDH1A1L3MBTL1PTGER3GPR55LMNA
SCHEMBL473945 0.85 ALDH1A1 (0.38) ALDH1A1L3MBTL1PTGER3USP30GPR55
SCHEMBL12163862 0.85 ALDH1A1 (0.38) ALDH1A1L3MBTL1PTGER3USP30GPR55
SCHEMBL474375 0.84 ALDH1A1 (0.37) ALDH1A1LMNANR1H2NR1H3RIPK1
SCHEMBL474474 0.83 GPR55 (0.37) ALDH1A1PTGER3GPR55LMNAPDE3B
SCHEMBL12163784 0.83 GPR55 (0.37) ALDH1A1PTGER3GPR55LMNAPDE3B
SCHEMBL12163808 0.83 GPR55 (0.37) ALDH1A1PTGER3GPR55PDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-A1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed