SCHEMBL4740733

SCHEMBL4740733

CC1CC2(CCN1CC1CCC1)C(NC1CCCCC1)=NC(=O)N2c1cccc(Br)c1

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.35
HPGD P15428 1/20 0.35
RORC P51449 1/20 0.34
OPRD1 P41143 5/20 0.32
OPRM1 P35372 4/20 0.32
OPRK1 P41145 4/20 0.32
OPRL1 P41146 2/20 0.32
MEN1 O00255 1/20 0.32
ADORA3 P0DMS8 2/20 0.31
ADORA1 P30542 2/20 0.31
HSP90AA1 P07900 1/20 0.30
MAPT P10636 1/20 0.30
THRB P10828 1/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL755089 1.00 KMT2A (0.35) KMT2AHPGDRORCOPRD1OPRM1
Hydrochloric Acid SCHEMBL5616268 0.99 KMT2A (0.34) KMT2AHPGDRORCOPRD1OPRM1
Hydrochloric Acid SCHEMBL757174 0.99 KMT2A (0.34) KMT2AHPGDRORCOPRD1OPRM1
SCHEMBL757090 0.91 MAPT (0.36) KMT2AHPGDOPRD1OPRM1OPRK1
SCHEMBL757580 0.91 MAPT (0.36) KMT2AHPGDOPRD1OPRM1OPRK1
Hydrochloric Acid SCHEMBL755877 0.90 MAPT (0.35) KMT2AHPGDOPRD1OPRM1OPRK1
SCHEMBL764691 0.89 ADORA3 (0.40) OPRD1OPRM1OPRK1OPRL1ADORA3
SCHEMBL755429 0.80 BACE1 (0.34) OPRD1OPRM1OPRL1ADORA3ADORA1
SCHEMBL760030 0.80 BACE1 (0.34) OPRD1OPRM1OPRL1ADORA3ADORA1
SCHEMBL755862 0.80 BACE1 (0.34) OPRD1OPRM1OPRL1ADORA3ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910364-A2 SPIROPIPERIDINE BETA-SECRETASE INHIBITORS FOR THE TREATMENT OF ALZHEIMER'S DISEASE Merck & Co., Inc. (US) 2008-04-16 EP claimed
WO-2007011833-A2 SPIROPIPERIDINE BETA-SECRETASE INHIBITORS FOR THE TREATMENT OF ALZHEIMER'S DISEASE MERCK & CO., INC. (US) 2007-01-25 WO claimed
WO-2007011810-A1 SPIROPIPERIDINE BETA-SECRETASE INHIBITORS FOR THE TREATMENT OF ALZHEIMER'S DISEASE MERCK & CO., INC. (US) 2007-01-25 WO claimed