SCHEMBL4741585

SCHEMBL4741585

NC1(c2ccccc2)NC(=O)c2nc[nH]c2N1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.35
BACE1 P56817 1/20 0.35
BACE2 Q9Y5Z0 1/20 0.35
POLB P06746 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
KDM4E B2RXH2 3/20 0.34
MAPT P10636 2/20 0.34
CYP2C9 P11712 2/20 0.34
BLM P54132 2/20 0.34
PMP22 Q01453 2/20 0.34
CYP3A4 P08684 1/20 0.34
CACNA1F O60840 1/20 0.34
HTR2A P28223 1/20 0.34
HRH1 P35367 1/20 0.34
SCN1A P35498 1/20 0.34
SCN4A P35499 1/20 0.34
CACNA1D Q01668 1/20 0.34
KCNH2 Q12809 1/20 0.34
CACNA1S Q13698 1/20 0.34
CACNA1C Q13936 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1286941 0.79 FNTA (0.34) ALDH1A1POLBRXFP1KDM4EMAPT
SCHEMBL5958156 0.75 ABL1 (0.34) ALDH1A1BACE1POLBRXFP1KDM4E
SCHEMBL6536476 0.69 MEN1 (0.31) BLMKMT2A
SCHEMBL23648186 0.68 CYP1A2 (0.32)
SCHEMBL9662746 0.66 GDA (0.30)
SCHEMBL4267183 0.64
SCHEMBL13946583 0.57 KDM4E (0.54) ALDH1A1KDM4EMAPTCYP3A4LMNA
SCHEMBL23691776 0.57 ALDH1A1 (0.35) ALDH1A1POLBRXFP1BLMKMT2A
SCHEMBL6425456 0.57 CYP2C9 (0.59) ALDH1A1BACE1BACE2MAPTCYP2C9
SCHEMBL30464742 0.56 GSK3B (0.43) ALDH1A1BACE1BACE2POLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008094203-A2 POLAR ESTER PRODRUGS OF HETEROCYCLIC HYBRID ANTIBACTERIAL COMPOUNDS AND SALTS THEREOF MICROBIOTIX, INC. (US) 2008-08-07 WO disclosed